SCHEMBL3410075

SCHEMBL3410075

COc1nccc(-n2cccn2)c1C(=O)N(OC)c1cncnc1

nearest known ligand 0.37

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.37
CYP46A1 Q9Y6A2 1/20 0.36
KDM4E B2RXH2 3/20 0.36
CYP1A2 P05177 2/20 0.36
CYP2C19 P33261 2/20 0.36
CYP2D6 P10635 1/20 0.36
HCRTR1 O43613 5/20 0.35
MEN1 O00255 2/20 0.34
HPGD P15428 2/20 0.34
NPSR1 Q6W5P4 1/20 0.34
HCRTR2 O43614 4/20 0.33
EGLN1 Q9GZT9 3/20 0.33
KCNH2 Q12809 1/20 0.33
ALDH1A1 P00352 1/20 0.33
MAPT P10636 1/20 0.33
LMNA P02545 1/20 0.33
EGFR P00533 1/20 0.32
ATR Q13535 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3408373 0.84 HCRTR1 (0.34) KMT2ACYP46A1KDM4ECYP1A2CYP2C19
SCHEMBL3406965 0.77 HCRTR2 (0.47) KMT2AKDM4ECYP1A2CYP2C19CYP2D6
SCHEMBL3407758 0.71 LMNA (0.36) KMT2ACYP46A1KDM4ECYP1A2CYP2C19
SCHEMBL3406978 0.70 SQOR (0.33) KMT2ACYP46A1KDM4ECYP1A2CYP2C19
SCHEMBL3406972 0.70 ATR (0.37) KMT2ACYP46A1KDM4ECYP1A2CYP2C19
SCHEMBL3410082 0.68 MEN1 (0.35) KMT2ACYP46A1KDM4ECYP1A2CYP2C19
SCHEMBL26342753 0.66 NPC1 (0.45) KMT2AKDM4ECYP1A2CYP2C19CYP2D6
SCHEMBL3408377 0.65 SCN9A (0.34) KMT2AKDM4ECYP1A2CYP2C19CYP2D6
SCHEMBL9343163 0.65 CA12 (0.56) KMT2AKDM4ECYP1A2CYP2C19CYP2D6
SCHEMBL2900508 0.65 TRPV1 (0.45) KMT2ACYP46A1KDM4ECYP1A2CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010038081-A2 HETEROCYCLIC DERIVATIVES AND METHODS OF USE THEREOF ASTRAZENECA AB (SE) 2010-04-08 WO disclosed