SCHEMBL3433145

SCHEMBL3433145

COC(=O)c1ccc2cccc(O)c2n1.COC(=O)c1ccc2cccc(OS(=O)(=O)C(F)(F)F)c2n1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.49
KDM4E B2RXH2 3/20 0.49
PDE4D Q08499 2/20 0.46
PIM1 P11309 1/20 0.45
CA1 P00915 1/20 0.44
CA2 P00918 1/20 0.44
MMP2 P08253 1/20 0.39
PTGER4 P35408 1/20 0.37
MEN1 O00255 1/20 0.37
NPC1 O15118 1/20 0.37
RAB9A P51151 1/20 0.37
MAPT P10636 3/20 0.37
ALDH1A1 P00352 2/20 0.37
GLA P06280 1/20 0.37
HPGD P15428 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
HDAC3 O15379 1/20 0.37
HDAC4 P56524 1/20 0.37
HDAC1 Q13547 1/20 0.37
HDAC7 Q8WUI4 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2118060 0.95 CA1 (0.45) KMT2AKDM4EPDE4DCA1CA2
SCHEMBL3425983 0.84 MAPT (0.47) KMT2AKDM4EPDE4DPIM1MEN1
SCHEMBL847651 0.83 KDM4E (0.65) KMT2AKDM4EPDE4DPIM1CA1
SCHEMBL7362665 0.82 KMT2A (0.54) KMT2AKDM4EPDE4DPIM1CA1
SCHEMBL7362663 0.80 KDM4E (0.77) KMT2AKDM4EPDE4DPIM1CA1
SCHEMBL2116612 0.79 MAPT (0.50) KMT2AKDM4EMEN1MAPTALDH1A1
SCHEMBL2944266 0.78 METAP2 (0.40) KMT2AKDM4EPDE4DMETAP2
SCHEMBL4701058 0.76 KDM4E (0.56) KMT2AKDM4EPDE4DCA1CA2
SCHEMBL2950729 0.76 ALDH1A1 (0.44) KMT2AKDM4EPDE4DCA1CA2
SCHEMBL590594 0.75 MTNR1A (0.42) PDE4DCA1CA2METAP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2250152-A1 QUINOLINES AS INHIBITORS OF FARNESYL PYROPHOSPHATE SYNTHASE Novartis AG (CH) 2010-11-17 EP disclosed
WO-2009106586-A1 QUINOLINES AS INHIBITORS OF FARNESYL PYROPHOSPHATE SYNTHASE NOVARTIS AG (CH) 2009-09-03 WO disclosed