SCHEMBL3433646

SCHEMBL3433646

Nc1cc2ccc3ccccc3c2[nH]1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 8/20 0.53
HSD17B10 Q99714 6/20 0.53
HPGD P15428 4/20 0.53
MEN1 O00255 1/20 0.53
USP2 O75604 1/20 0.53
KMT2A Q03164 1/20 0.53
AOC3 Q16853 2/20 0.52
KIF11 P52732 1/20 0.47
KDM4E B2RXH2 2/20 0.44
RAB9A P51151 1/20 0.44
SIRT2 Q8IXJ6 1/20 0.44
SIRT1 Q96EB6 1/20 0.44
TSHR P16473 2/20 0.44
CYP2A6 P11509 2/20 0.44
TDP1 Q9NUW8 1/20 0.44
HPRT1 P00492 2/20 0.44
HTT P42858 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
HIF1A Q16665 1/20 0.43
CYP1B1 Q16678 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4417853 0.79 AOC3 (0.48) ALDH1A1HSD17B10AOC3CYP3A4
SCHEMBL28669933 0.77 ALDH1A1 (0.55) ALDH1A1HSD17B10HPGDMEN1USP2
SCHEMBL29275406 0.75 ALDH1A1 (0.53) ALDH1A1HSD17B10HPGDMEN1USP2
SCHEMBL4916031 0.75 ALDH1A1 (0.58) ALDH1A1HSD17B10HPGDMEN1USP2
SCHEMBL30494604 0.75 ALDH1A1 (0.53) ALDH1A1HSD17B10HPGDMEN1USP2
SCHEMBL7915531 0.75 ALDH1A1 (0.66) ALDH1A1HSD17B10HPGDMEN1USP2
SCHEMBL27085550 0.74 CYP3A4 (0.49) ALDH1A1HSD17B10MEN1KMT2AKDM4E
Iodide SCHEMBL27218977 0.73 ALDH1A1 (0.64) ALDH1A1HSD17B10HPGDMEN1USP2
SCHEMBL31020778 0.72 RAB9A (0.55) ALDH1A1HSD17B10HPGDMEN1USP2
SCHEMBL4891254 0.72 RAB9A (0.55) ALDH1A1HSD17B10HPGDMEN1USP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5498727-A Preparation of benzindole compounds from naphthalene compounds AGOURON PHARMACEUTICALS, INC. (US) 1996-03-12 US claimed
WO-1996002502-A1 PREPARATION OF BENZINDOLE COMPOUNDS FROM NAPHTHALENE COMPOUNDS AGOURON PHARMACEUTICALS, INC. (US) 1996-02-01 WO claimed
WO-2010027280-A1 NITROBENZINDOLES AND THEIR USE IN CANCER THERAPY AUCKLAND UNISERVICES LIMITED (NZ) 2010-03-11 WO disclosed