SCHEMBL3433756

SCHEMBL3433756

CC(c1ccccc1)c1cccc(-c2ccc3nccnc3c2)c1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TGFBR1 P36897 9/20 0.45
PSEN1 P49768 1/20 0.39
PSEN2 P49810 1/20 0.39
APH1B Q8WW43 1/20 0.39
NCSTN Q92542 1/20 0.39
APH1A Q96BI3 1/20 0.39
PSENEN Q9NZ42 1/20 0.39
PIK3CD O00329 1/20 0.39
RXRA P19793 1/20 0.39
RXRB P28702 1/20 0.39
RXRG P48443 1/20 0.39
FLT3 P36888 1/20 0.38
GSK3B P49841 1/20 0.38
ABCB1 P08183 1/20 0.37
ABCC1 P33527 1/20 0.37
ABCG2 Q9UNQ0 1/20 0.37
ATP1A1 P05023 1/20 0.37
ATP1B1 P05026 1/20 0.37
ATP1A3 P13637 1/20 0.37
ATP1B2 P14415 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3388523 0.83 BRD4 (0.49) TGFBR1RXRARXRBRXRG
SCHEMBL3418697 0.81 TGFBR1 (0.42) TGFBR1FLT3GSK3BPIK3CA
SCHEMBL27906803 0.79 TGFBR1 (0.53) TGFBR1PIK3CDFLT3GSK3BABCB1
SCHEMBL3433216 0.77 PSEN1 (0.46) TGFBR1PSEN1PSEN2APH1BNCSTN
SCHEMBL24686234 0.76 TGFBR1 (0.50) TGFBR1PIK3CDFLT3GSK3BABCB1
SCHEMBL8337311 0.73 NPC1 (0.52) TGFBR1FLT3GSK3B
SCHEMBL21508010 0.73 OGA (0.41) TGFBR1PIK3CDPIK3CA
SCHEMBL3390623 0.71 ALK (0.55) TGFBR1GSK3BABCB1ABCC1ABCG2
SCHEMBL2210935 0.71 TYR (0.47)
Tannin Pyrogallol SCHEMBL29187614 0.71 PTGS2 (0.52) RXRARXRBRXRG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010052448-A2 FUSED PYRAZINE DERIVATIVES AS KINASE INHIBITORS UCB PHARMA S.A. (BE) 2010-05-14 WO disclosed