SCHEMBL3434283

SCHEMBL3434283

NC(=O)C1CCCN(c2ncc[nH]2)C1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PBK Q96KB5 1/20 0.58
LRRK2 Q5S007 2/20 0.47
HSD17B10 Q99714 3/20 0.43
KDM4E B2RXH2 3/20 0.43
ALDH1A1 P00352 2/20 0.43
HPGD P15428 1/20 0.43
PRKDC P78527 1/20 0.41
EIF2AK4 Q9P2K8 3/20 0.41
JAK2 O60674 2/20 0.41
JAK3 P52333 2/20 0.41
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
OPRM1 P35372 1/20 0.40
OPRD1 P41143 1/20 0.40
OPRK1 P41145 1/20 0.40
OGFRL1 Q5TC84 1/20 0.40
CDK9 P50750 1/20 0.40
GLA P06280 1/20 0.39
GAA P10253 1/20 0.39
ATR Q13535 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29952582 0.74 HIPK2 (0.35) PBKJAK3
SCHEMBL8235149 0.74 PBK (1.00) PBKLRRK2JAK2JAK3ATR
SCHEMBL18395530 0.72 KMT2A (0.61) PBKKDM4EKMT2A
SCHEMBL3955342 0.72 PBK (0.70) PBKLRRK2PRKDCJAK2JAK3
SCHEMBL1290812 0.71 GPBAR1 (0.57) PBKLRRK2HSD17B10KDM4EALDH1A1
SCHEMBL556899 0.71 LMNA (0.39)
SCHEMBL300491 0.71 ALOX15 (0.41) HSD17B10KDM4EALDH1A1HPGDJAK3
SCHEMBL311710 0.69 BCHE (0.42) ALDH1A1HPGDJAK2JAK3MEN1
Hydrochloric Acid SCHEMBL9200760 0.69 ALOX15 (0.39) KDM4EALDH1A1HPGDJAK3
SCHEMBL6820246 0.69 EIF2AK4 (0.60) PBKHSD17B10KDM4EALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2229363-A1 RENIN INHIBITORS Merck Frosst Canada Ltd. (CA) 2010-09-22 EP disclosed
WO-2009070869-A1 RENIN INHIBITORS MERCK FROSST CANADA LTD. (CA) 2009-06-11 WO disclosed