SCHEMBL3434306

SCHEMBL3434306

CC1(C)Nc2ccc(-c3ccc(OC(F)(F)F)cc3)cc2NC1=O

nearest known ligand 0.49

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ABL1 P00519 6/20 0.44
MMP2 P08253 5/20 0.43
MMP9 P14780 4/20 0.43
MMP8 P22894 1/20 0.43
CES1 P23141 1/20 0.43
SCN9A Q15858 1/20 0.41
NOTUM Q6P988 1/20 0.41
SCN5A Q14524 1/20 0.40
KIF11 P52732 1/20 0.40
MMP1 P03956 3/20 0.39
ADAMTS5 Q9UNA0 1/20 0.39
MMP3 P08254 2/20 0.39
CA12 O43570 1/20 0.38
CA9 Q16790 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3433509 0.88 OTUD7B (0.48) ABL1CES1SCN9AADAMTS5
SCHEMBL1897022 0.70 GRIA1 (0.60) CES1NOTUMKIF11
SCHEMBL22314930 0.70 CES1 (0.64) ABL1CES1
SCHEMBL2264074 0.70 CES1 (0.51) CES1ADAMTS5
SCHEMBL14499205 0.69 PGR (0.42) CA9
SCHEMBL3310995 0.69 KIF11 (0.70) CES1KIF11
SCHEMBL7170898 0.68 CSNK1G1 (0.45) ADAMTS5CA12CA9
SCHEMBL3596379 0.68 MGAT2 (0.37)
SCHEMBL13717944 0.68 ABL1 (0.52) ABL1CA12CA9
SCHEMBL941821 0.68 MMP2 (0.49) MMP2MMP9MMP8SCN9ANOTUM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010053757-A1 2 -OXOQUINOXALIN BLOCKERS OF THE LATE SODIUM CHANNEL GILEAD PALO ALTO, INC. (US) 2010-05-14 WO claimed