SCHEMBL3434604

SCHEMBL3434604

COc1cc(C)[c]c(O)c1OCCCc1ccccc1

nearest known ligand 0.48

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ADRB2 P07550 1/20 0.45
DRD2 P14416 1/20 0.45
DRD1 P21728 1/20 0.45
DRD4 P21917 1/20 0.45
DRD3 P35462 1/20 0.45
ALOX5 P09917 2/20 0.44
SCN9A Q15858 1/20 0.44
AKR1B10 O60218 1/20 0.41
AKR1B1 P15121 1/20 0.41
TRPV1 Q8NER1 1/20 0.41
PDE4A P27815 1/20 0.41
PDE4B Q07343 1/20 0.41
PDE4C Q08493 1/20 0.41
PDE4D Q08499 1/20 0.41
NPC1 O15118 1/20 0.41
RAB9A P51151 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3386404 0.87 SMN1; SMN2 (0.41) ADRB2DRD2DRD1DRD4DRD3
SCHEMBL3762438 0.75 ALOX5 (0.50) ALOX5SCN9AAKR1B10AKR1B1TRPV1
SCHEMBL1541828 0.75 SMN1; SMN2 (0.47) SCN9APDE4D
SCHEMBL1542014 0.72 PDE4D (0.48) ALOX5SCN9AAKR1B10AKR1B1TRPV1
SCHEMBL14835642 0.71 ALOX5 (0.51) ALOX5SCN9ANPC1RAB9A
SCHEMBL13339111 0.71 MAPT (0.48)
SCHEMBL1541630 0.70 IDO1 (0.40) ADRB2DRD2DRD1DRD4DRD3
SCHEMBL1541608 0.70 PDE4D (0.51) ALOX5SCN9APDE4APDE4BPDE4C
SCHEMBL11419578 0.70 HTR1A (0.58) ADRB2DRD2DRD1DRD4DRD3
SCHEMBL7896500 0.69 TUBB4A (0.61)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2197832-A1 NOVEL ARYL POTASSIUM CHANNEL BLOCKERS AND USES THEREOF Bionomics Limited (AU) 2010-06-23 EP disclosed
WO-2009043117-A1 NOVEL ARYL POTASSIUM CHANNEL BLOCKERS AND USES THEREOF BIONOMICS LIMITED (AU) 2009-04-09 WO disclosed