Neostigmine

Neostigmine

SCHEMBL34419

CN(C)C(=O)Oc1cccc([N+](C)(C)C)c1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ACHE

The experimentally established mechanism targets of Neostigmine. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ACHE known ✓ P22303 13/20 1.00
BCHE P06276 7/20 1.00
LMNA P02545 4/20 1.00
MEN1 O00255 1/20 0.97
KMT2A Q03164 1/20 0.97
NPSR1 Q6W5P4 1/20 0.97
RAB9A P51151 1/20 0.53
GLA P06280 2/20 0.47
TSHR P16473 1/20 0.47
MAPK1 P28482 1/20 0.47
NCEH1 Q6PIU2 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Neostigmine SCHEMBL29603805 1.00 ACHE (1.00) ACHEBCHELMNAMEN1KMT2A
Neostigmine SCHEMBL8026154 1.00 ACHE (1.00) ACHEBCHELMNAMEN1KMT2A
Neostigmine SCHEMBL29618009 0.98 ACHE (1.00) ACHEBCHELMNAMEN1KMT2A
Neostigmine SCHEMBL30029632 0.98 ACHE (0.97) ACHEBCHELMNAMEN1KMT2A
Neostigmine SCHEMBL20425365 0.98 ACHE (0.97) ACHEBCHELMNAMEN1KMT2A
Neostigmine SCHEMBL41128 0.98 ACHE (1.00) ACHEBCHELMNAMEN1KMT2A
Neostigmine SCHEMBL16228482 0.98 ACHE (0.97) ACHEBCHELMNAMEN1KMT2A
Neostigmine SCHEMBL7576189 0.97 ACHE (0.94) ACHEBCHELMNAMEN1KMT2A
Neostigmine SCHEMBL7633009 0.94 ACHE (0.88) ACHEBCHELMNAMEN1KMT2A
Neostigmine SCHEMBL2028206 0.93 ACHE (0.89) ACHEBCHELMNAMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 10473 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3607938-B1 PHARMACEUTICAL COMPOSITION SOVIC BRKICIC LJILJANA (HR) 2026-05-27 EP claimed
CN-224242693-U Novel stigmine injection split charging structure of glycopyrronium bromide 广州曼翔医药有限公司 2026-05-15 CN claimed
EP-4736841-A1 A MUCOADHESIVE LAYER FOR BUCCAL ADMINISTRATION OF AN ACTIVE PHARMACEUTICAL INGREDIENT IQ medical GmbH (DE) 2026-05-06 EP claimed
EP-4665351-A1 IMPROVING GLYMPHATIC-LYMPHATIC EFFLUX University of Rochester (US) 2025-12-24 EP claimed
US-20250375373-A1 READY-TO-USE INJECTABLE PHARMACEUTICAL COMPOSITIONS COMPRISING NEOSTIGMINE AND GLYCOPYRROLATE AZURITY PHARMACEUTICALS, INC. (US) 2025-12-11 US claimed
EP-4635489-A1 COMPOSITION FOR PREVENTING OR TREATING SIDE EFFECTS OF CHOLINESTERASE INHIBITORS Dr.Noah Biotech Inc. (KR) 2025-10-22 EP claimed
US-12403262-B2 Tamper evident assembly with RFID for syringes FRESENIUS KABI USA, LLC (US) 2025-09-02 US claimed
US-12390454-B2 Use and composition for protection against organophosphorus poisoning CLARENCE SMITH KATHLEEN E (US) 2025-08-19 US claimed
US-12383491-B2 Ready-to-use injectable pharmaceutical compositions comprising neostigmine and glycopyrrolate AZURITY PHARMACEUTICALS, INC. (US) 2025-08-12 US claimed
US-20250249185-A1 TAMPER EVIDENT CAP WITH RFID FOR SYRINGES FRESENIUS KABI USA, LLC 2025-08-07 US claimed
US-4736024-A Process for preparing salt of hyaluronic acid with a pharmaceutically active substance FIDIA, S.P.A. (IT) 1988-04-05 US claimed
US-4661509-A ENZYME INHIBITORS GORDON ARNOLD Z 1987-04-28 US claimed
EP-0197718-A2 New medicaments for topical use FIDIA S.p.A. (IT) 1986-10-15 EP claimed
US-4590166-A WASHING WITH WATER AND ALCOHOL THE UNITED STATES OF AMERICA AS REPRESENTED BY THE SECRETARY OF THE ARMY (US) 1986-05-20 US claimed
US-4562196-A ANTAGONIST OF MUSCLE RELAXANTS NELSON RESEARCH & DEVELOPMENT (US) 1985-12-31 US claimed
EP-0152379-A2 Process for preparing pharmaceutical compositions containing unilamellar liposomes CIBA-GEIGY AG (CH) 1985-08-21 EP claimed
EP-0126684-A2 Drug delivery system utilizing thermosetting gels MERCK & CO. INC. (US) 1984-11-28 EP claimed
US-4474751-A SUSTAINED RELEASE USING AN ALKYLENEDIAMINE-MODIFIED ETHYLENE OXIDE-PROPYLENE OXIDE COPOLYMER MERCK & CO., INC. (US) 1984-10-02 US claimed
US-4439427-A Method and composition for treating pediculosis SOFT SHEEN PRODUCTS, INC. (US) 1984-03-27 US claimed
EP-0001924-B1 PHARMACEUTICAL COMPOSITION FOR ADMINISTERING CHOLINE MASSACHUSETTS INSTITUTE OF TECHNOLOGY (US) 1982-07-07 EP claimed