Neostigmine

Neostigmine

SCHEMBL41128

CN(C)C(=O)Oc1cccc([N+](C)(C)C)c1.[Br-]

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ACHE

The experimentally established mechanism targets of Neostigmine. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ACHE known ✓ P22303 14/20 1.00
BCHE P06276 6/20 1.00
LMNA P02545 4/20 1.00
MEN1 O00255 1/20 1.00
KMT2A Q03164 1/20 1.00
NPSR1 Q6W5P4 1/20 1.00
RAB9A P51151 1/20 0.52
GLA P06280 2/20 0.49
TSHR P16473 1/20 0.46
MAPK1 P28482 1/20 0.46
NCEH1 Q6PIU2 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Neostigmine SCHEMBL29618009 1.00 ACHE (1.00) ACHEBCHELMNAMEN1KMT2A
Neostigmine SCHEMBL8026154 0.98 ACHE (1.00) ACHEBCHELMNAMEN1KMT2A
Neostigmine SCHEMBL29603805 0.98 ACHE (1.00) ACHEBCHELMNAMEN1KMT2A
Neostigmine SCHEMBL34419 0.98 ACHE (1.00) ACHEBCHELMNAMEN1KMT2A
Neostigmine SCHEMBL20425365 0.97 ACHE (0.97) ACHEBCHELMNAMEN1KMT2A
Neostigmine SCHEMBL16228482 0.97 ACHE (0.97) ACHEBCHELMNAMEN1KMT2A
Neostigmine SCHEMBL30029632 0.97 ACHE (0.97) ACHEBCHELMNAMEN1KMT2A
Neostigmine SCHEMBL7576189 0.95 ACHE (0.94) ACHEBCHELMNAMEN1KMT2A
Neostigmine SCHEMBL21772308 0.94 ACHE (0.89) ACHEBCHELMNAMEN1KMT2A
Neostigmine SCHEMBL2028206 0.94 ACHE (0.89) ACHEBCHELMNAMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 2294 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12292363-B2 Method for preparing biological material having excellent light-transmitting property RIKEN (JP) 2025-05-06 US claimed
CN-119894225-A Perovskite active layer film based on neostigmine bromide passivator, and preparation method and application thereof 常州大学 2025-04-25 CN claimed
CN-118258926-A Method for detecting glycopyrronium bromide isomer in glycopyrronium bromide neostigmine injection and quality control standard thereof 北京阜康仁生物制药科技有限公司 2024-06-28 CN claimed
CN-117357476-A New stigmine glycopyrrolate injection and preparation method thereof 李宏 2024-01-09 CN claimed
CN-113277961-B Synthesis method of bromneostigmine 深圳市新浩瑞医药科技有限公司 2023-05-09 CN claimed
WO-2023059810-A1 STENTS AND METHODS OF USE UNIVERSITY OF CONNECTICUT (US) 2023-04-13 WO claimed
WO-2023044463-A1 SILK FIBROIN DERIVED BRUSH-LIKE POLYMERS UNIVERSITY OF CONNECTICUT (US) 2023-03-23 WO claimed
US-20220381657-A1 METHOD FOR PREPARING BIOLOGICAL MATERIAL HAVING EXCELLENT LIGHT-TRANSMITTING PROPERTY RIKEN (JP) 2022-12-01 US claimed
US-11389420-B2 Pharmaceutical compositions and methods utilizing neostigmine and an NK-1 antagonist for treating myasthenia gravis DAS-MG, INC. (US) 2022-07-19 US claimed
CN-113358528-B Method for detecting acetylcholinesterase and inhibitor thereof based on pendant drop method 山东大学 2022-06-17 CN claimed
WO-2000074655-A2 DELAYED TOTAL RELEASE TWO PULSE GASTROINTESTINAL DRUG DELIVERY SYSTEM DEXCEL PHARMA TECHNOLOGIES LTD. (IL) 2000-12-14 WO claimed
CN-1274280-A Delayed total release gastrointestinal delivery system PERIO PROD LTD (IL) 2000-11-22 CN claimed
EP-1021171-A1 DELAYED TOTAL RELEASE GASTROINTESTINAL DRUG DELIVERY SYSTEM Perio Products Ltd (IL) 2000-07-26 EP claimed
WO-1999018938-A1 DELAYED TOTAL RELEASE GASTROINTESTINAL DRUG DELIVERY SYSTEM PERIO PRODUCTS LTD. (IL) 1999-04-22 WO claimed
EP-0166724-B1 COMPOSITION FOR TREATING PEDICULOSIS SOFT SHEEN PRODUCTS, INC. (US) 1990-11-22 EP claimed
EP-0166724-A1 COMPOSITION FOR TREATING PEDICULOSIS. SOFT SHEEN PRODUCTS INC (US) 1986-01-08 EP claimed
WO-1985002755-A1 METHOD AND COMPOSITION FOR TREATING PEDICULOSIS SOFT SHEEN PRODUCTS, INC. (US) 1985-07-04 WO claimed
EP-0140434-A2 Pharmaceutical composition with systemic anticholineesterasic, agonistic-cholinergic and antimuscarinic activity PRODOTTI FORMENTI S.r.l. (IT) 1985-05-08 EP claimed
US-4439427-A Method and composition for treating pediculosis SOFT SHEEN PRODUCTS, INC. (US) 1984-03-27 US claimed
US-4098899-A NEOSTIGMINE BROMIDE OR NEOSTIGMINE METHYL SULFATE SCHWARTZ GEORGE R 1978-07-04 US claimed