SCHEMBL3453136

SCHEMBL3453136

NC(=O)c1c(O)ccc(-c2ccccc2)c1C(N)=O

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BCAT2 O15382 2/20 0.50
BACE1 P56817 2/20 0.45
ALOX5 P09917 1/20 0.44
ALDH1A1 P00352 3/20 0.43
HPGD P15428 3/20 0.43
HSD17B10 Q99714 3/20 0.43
BCL2L1 Q07817 1/20 0.43
LMNA P02545 2/20 0.43
MAPT P10636 2/20 0.41
TSHR P16473 2/20 0.41
KDM4E B2RXH2 1/20 0.41
POLB P06746 1/20 0.40
CYP3A4 P08684 1/20 0.40
PARP1 P09874 1/20 0.40
CYP2C19 P33261 1/20 0.40
RECQL P46063 1/20 0.40
BLM P54132 1/20 0.40
PMP22 Q01453 1/20 0.40
TDP1 Q9NUW8 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL975812 0.85 BCAT2 (0.55) BCAT2BACE1ALDH1A1HPGDHSD17B10
SCHEMBL27967445 0.83 BCAT2 (0.42) BCAT2BACE1ALOX5ALDH1A1HPGD
SCHEMBL4881197 0.81 BCAT2 (0.60) BCAT2ALDH1A1HPGDHSD17B10MAPT
SCHEMBL28429428 0.80 CA12 (0.52) BACE1ALOX5ALDH1A1HPGDHSD17B10
SCHEMBL6842022 0.79 BCAT2 (0.63) BCAT2ALDH1A1HPGDHSD17B10BCL2L1
SCHEMBL2000711 0.78 HSD17B10 (0.46) ALDH1A1HPGDHSD17B10MAPTTSHR
SCHEMBL5590480 0.74 HNF4A (0.48) BACE1ALOX5ALDH1A1HPGDHSD17B10
SCHEMBL27718034 0.74 HNF4A (0.53) BACE1ALOX5ALDH1A1HPGDHSD17B10
SCHEMBL722165 0.74 BCAT2 (0.47) BCAT2ALDH1A1HPGDHSD17B10MAPT
SCHEMBL4143761 0.74 BCAT2 (0.56) BCAT2ALDH1A1HPGDHSD17B10MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2205070-A1 N-HYDROXY-NAPHTHALENE DICARBOXAMIDE AND N-HYDROXY-BIPHENYL-DICARBOXAMIDE COMPOUNDS AS HISTONE DEACETYLASE INHIBITORS Merck Sharp & Dohme Corp. (US) 2010-07-14 EP disclosed
WO-2009045385-A1 N-HYDROXY-NAPHTHALENE DICARBOXAMIDE AND N-HYDROXY-BIPHENYL-DICARBOXAMIDE COMPOUNDS AS HISTONE DEACETYLASE INHIBITORS MERCK & CO., INC. (US) 2009-04-09 WO disclosed