SCHEMBL3464148

SCHEMBL3464148

Cc1ccc(S(=O)(=O)n2cc(Br)cc2[CH]CC(N)=O)cc1

nearest known ligand 0.40

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.40
CA1 P00915 1/20 0.40
CA2 P00918 1/20 0.40
NOD2 Q9HC29 1/20 0.37
NOD1 Q9Y239 1/20 0.37
RAPGEF4 Q8WZA2 1/20 0.36
L3MBTL1 Q9Y468 2/20 0.36
KDM4E B2RXH2 2/20 0.36
UBE2N P61088 1/20 0.36
HTR6 P50406 1/20 0.36
THRB P10828 1/20 0.36
LMNA P02545 1/20 0.35
TSHR P16473 1/20 0.35
HDAC1 Q13547 1/20 0.35
ALK Q9UM73 1/20 0.35
KMT2A Q03164 1/20 0.34
MAPT P10636 1/20 0.34
EGFR P00533 1/20 0.34
ERBB2 P04626 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL568356 0.85 ALDH1A1 (0.40) ALDH1A1CA1CA2NOD2NOD1
SCHEMBL8514020 0.83 ALDH1A1 (0.40) ALDH1A1CA1CA2NOD2NOD1
SCHEMBL4170909 0.79 KDM4E (0.49) ALDH1A1CA1CA2NOD1RAPGEF4
SCHEMBL29564645 0.73 CA1 (0.42) ALDH1A1CA1CA2NOD1RAPGEF4
SCHEMBL10004099 0.72 NOD2 (0.54) ALDH1A1CA1CA2NOD2NOD1
SCHEMBL22689649 0.72 FBP1 (0.44) CA1CA2NOD1RAPGEF4L3MBTL1
SCHEMBL22689650 0.72 FBP1 (0.44) CA1CA2NOD1RAPGEF4L3MBTL1
SCHEMBL2184458 0.72 CA1 (0.43) ALDH1A1CA1CA2NOD2NOD1
SCHEMBL568306 0.71 CA1 (0.45) ALDH1A1CA1CA2NOD2NOD1
SCHEMBL10003393 0.71 CA1 (0.40) CA1CA2NOD2NOD1RAPGEF4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2346868-B1 AZAINDAZOLE COMPOUNDS AS CCR1 RECEPTOR ANTAGONISTS BOEHRINGER INGELHEIM INT (DE) 2016-01-27 EP disclosed
US-8338610-B2 Pyridinyl compounds useful as intermediates BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2012-12-25 US disclosed
US-20120136158-A1 Pyridinyl Compounds Useful As Intermediates BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2012-05-31 US disclosed
US-20100093724-A1 Azaindazole Compounds As CCR1 Receptor Antagonists BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2010-04-15 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100093724-A1 Azaindazole Compounds As CCR1 Receptor Antagonists CCR1, CCR3, CCR4 ALDH1A1 523/4885CA1 1081/4885CA2 2686/4885
US-20120136158-A1 Pyridinyl Compounds Useful As Intermediates CCR1, CCRL2, CCR4 ALDH1A1 268/4885CA1 2206/4885CA2 3968/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.