SCHEMBL3466804

SCHEMBL3466804

CC(=O)OC1Cc2cc(-c3ccc(Cl)cc3)ccc2NC1=O

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PGR P06401 4/20 0.40
TDP2 O95551 1/20 0.39
AHR P35869 1/20 0.38
JAK2 O60674 1/20 0.37
NTRK1 P04629 1/20 0.37
MET P08581 1/20 0.37
FGFR1 P11362 1/20 0.37
PRKACA P17612 1/20 0.37
KDR P35968 1/20 0.37
MAP2K2 P36507 1/20 0.37
FLT3 P36888 1/20 0.37
GSK3B P49841 1/20 0.37
MAP2K1 Q02750 1/20 0.37
MST1R Q04912 1/20 0.37
NTRK3 Q16288 1/20 0.37
NTRK2 Q16620 1/20 0.37
CAMK1D Q8IU85 1/20 0.37
PDE3B Q13370 1/20 0.37
PDE3A Q14432 1/20 0.37
DRD2 P14416 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3467796 0.87 PGR (0.41) PGRTDP2NTRK1FLT3GSK3B
SCHEMBL3466901 0.74 PGR (0.41) PGRTDP2AHRJAK2NTRK1
SCHEMBL7212449 0.73 ESR2 (0.42) MEN1ALDH1A1KMT2AMAPK1LMNA
SCHEMBL10352638 0.72 CHRM1 (0.36) MAPK1
SCHEMBL1900155 0.68 AHR (0.77) PGRTDP2AHRPDE3BPDE3A
SCHEMBL19899024 0.67 NOTUM (0.39) DRD2DRD4
SCHEMBL29073339 0.67 BRD4 (0.40) TDP2AHRMEN1KMT2AMAPK1
SCHEMBL57232 0.66 MAP3K14 (0.39) MEN1KMT2ALMNA
SCHEMBL7866698 0.66 AHR (0.53) PGRAHRDRD2DRD4MEN1
SCHEMBL3307966 0.66 KIF11 (0.68) PGRTDP2AHRJAK2NTRK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010074807-A1 3, 4-DIHYDROQUINOLIN-2 ( 1H ) -ONE DERIVATIVES AS SODIUM CHANNEL MODULATORS GILEAD PALO ALTO, INC. (US) 2010-07-01 WO disclosed