SCHEMBL3467211

SCHEMBL3467211

O=C1Nc2cc(I)ccc2C1=O

nearest known ligand 0.71

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CES1 P23141 6/20 0.71
TGM2 P21980 6/20 0.71
MAOA P21397 7/20 0.55
MAOB P27338 7/20 0.55
TDP2 O95551 2/20 0.46
BCHE P06276 1/20 0.43
CA12 O43570 1/20 0.42
CA1 P00915 1/20 0.42
CA2 P00918 1/20 0.42
CA9 Q16790 1/20 0.42
ALDH1A1 P00352 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
5-Iodoisatin SCHEMBL75159 0.83 TGM2 (1.00) CES1TGM2MAOAMAOBCA12
5-Iodoisatin SCHEMBL30794223 0.83 TGM2 (1.00) CES1TGM2MAOAMAOBCA12
5-Iodoisatin SCHEMBL1482216 0.82 TGM2 (0.96) CES1TGM2MAOAMAOBCA12
5-Iodoisatin SCHEMBL28515786 0.82 TGM2 (0.96) CES1TGM2MAOAMAOBCA12
SCHEMBL22300581 0.77 MAOA (0.50) CES1TGM2MAOAMAOB
SCHEMBL4192180 0.77 CES1 (0.62) CES1TGM2MAOAMAOBBCHE
SCHEMBL30398896 0.77 CES1 (0.62) CES1TGM2MAOAMAOBBCHE
SCHEMBL8557 0.75 CES1 (0.71) CES1TGM2MAOAMAOBTDP2
SCHEMBL13564440 0.75 CES1 (0.60) CES1TGM2MAOAMAOBBCHE
SCHEMBL29494851 0.75 CES1 (1.00) CES1TGM2MAOAMAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 38 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111574426-B Diamine monomer containing isoindigo structure and black polyimide synthesized by diamine monomer 湘潭大学 2023-06-23 CN claimed
CN-115716795-A Donor-acceptor type compound based on isoindigo derivative, preparation method, molecular lead and molecular electric switch 华东理工大学 2023-02-28 CN claimed
CN-108431209-B Derived and mature hepatocyte types of liver stem cells and uses thereof 新加坡科技研究局 2023-02-10 CN claimed
CN-113912609-A Preparation method of natural alkaloid tryptanthrin and derivative thereof 江苏大学 2022-01-11 CN claimed
CN-111574426-A Diamine monomer containing isoindigo structure and black polyimide synthesized from diamine monomer 湘潭大学 2020-08-25 CN claimed
CN-102690226-A Multi-nitrogen substituted isatin derivative and synthetic method of multi-nitrogen substituted isatin derivative UNIV GUANGDONG TECHNOLOGY 2012-09-26 CN claimed
CN-113912609-B Preparation method of natural alkaloid tryptanthrin and derivatives thereof 江苏大学 2024-01-05 CN disclosed
CN-115716795-A Donor-acceptor type compound based on isoindigo derivative, preparation method, molecular lead and molecular electric switch 华东理工大学 2023-02-28 CN disclosed
CN-108431209-B Derived and mature hepatocyte types of liver stem cells and uses thereof 新加坡科技研究局 2023-02-10 CN disclosed
EP-4108659-A1 NOVEL HETEROCYCLIC DERIVATIVES USEFUL AS SHP2 INHIBITORS Jacobio Pharmaceuticals Co., Ltd. (CN) 2022-12-28 EP disclosed
CN-114539273-A Novel heterocyclic derivatives useful as SHP2 inhibitors 北京加科思新药研发有限公司 2022-05-27 CN disclosed
CN-109311848-B Novel heterocyclic derivatives useful as SHP2 inhibitors 北京加科思新药研发有限公司 2022-02-01 CN disclosed
CN-113912609-A Preparation method of natural alkaloid tryptanthrin and derivative thereof 江苏大学 2022-01-11 CN disclosed
US-5604227-A EXCITATORY AMINO ACID ANTAGONIST; MONO, DI OR TRI-ACETYLATION OR ALKYLATION IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1997-02-18 US disclosed
US-5602169-A USEFUL IN REDUCING NEURONAL DAMAGE DURING ISCHEMIC STROKE BRISTOL-MYERS SQUIBB COMPANY (US) 1997-02-11 US disclosed
US-5599814-A SUBSTITUTED PYRIDAZINO(4,5-B)QUINOLINES AS ANTAGONISTS OF EXCITATORY AMINO ACIDS IMPERIAL CHEMICAL INDUSTRIES, PLC (GB) 1997-02-04 US disclosed
EP-0747354-A1 3-Substituted oxindole derivatives as potassium channel modulators BRISTOL-MYERS SQUIBB COMPANY (US) 1996-12-11 EP disclosed
EP-0516297-B1 Pyridazinediones and their use in the treatment of neurological disorders ZENECA LTD (GB) 1996-10-30 EP disclosed
US-5565483-A ADMINISTERING AS THERAPY FOR ISCHEMIA, CONVULSIONS OR ASTHMA BRISTOL-MYERS SQUIBB COMPANY (US) 1996-10-15 US disclosed
EP-0516297-A1 Pyridazinediones and their use in the treatment of neurological disorders ZENECA LIMITED (GB) 1992-12-02 EP disclosed