5-Iodoisatin

5-Iodoisatin

SCHEMBL28515786

C.O=C1Nc2ccc(I)cc2C1=O

nearest known ligand 0.96

Full drug profile on Sugi Atlas →

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
TGM2 P21980 5/20 0.96
CES1 P23141 5/20 0.96
MAOA P21397 6/20 0.53
MAOB P27338 6/20 0.53
CA12 O43570 1/20 0.53
CA1 P00915 1/20 0.53
CA2 P00918 1/20 0.53
CA9 Q16790 1/20 0.53
ALDH1A1 P00352 1/20 0.53
CAPN9 O14815 1/20 0.51
CASP3 P42574 1/20 0.51
PDE3B Q13370 1/20 0.50
PDE3A Q14432 1/20 0.50
LRRK2 Q5S007 1/20 0.48
APP P05067 2/20 0.47
MAPT P10636 2/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
5-Iodoisatin SCHEMBL75159 0.98 TGM2 (1.00) TGM2CES1MAOAMAOBCA12
5-Iodoisatin SCHEMBL30794223 0.98 TGM2 (1.00) TGM2CES1MAOAMAOBCA12
5-Iodoisatin SCHEMBL1482216 0.96 TGM2 (0.96) TGM2CES1MAOAMAOBCA12
SCHEMBL7791509 0.85 TGM2 (0.77) TGM2CES1LRRK2APPMAPT
SCHEMBL3467211 0.82 CES1 (0.71) TGM2CES1MAOAMAOBCA12
SCHEMBL20682550 0.78 TGM2 (0.67) TGM2CES1MAOAMAOBLRRK2
5-Fluoroisatin SCHEMBL28512324 0.76 MAOB (0.59) TGM2CES1MAOAMAOBCA12
Methane SCHEMBL27958656 0.76 TGM2 (0.96) TGM2CES1MAOAMAOBCA12
Methane SCHEMBL28522344 0.76 TGM2 (0.96) TGM2CES1MAOAMAOBCA12
SCHEMBL29657257 0.75 ROS1 (0.67) TGM2CES1MAOAMAOBCA12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109384769-B Synthetic method of R-configuration 3-substituted-3-hydroxy oxindole compound 陕西师范大学 2020-12-22 CN claimed
CN-109384769-B Synthetic method of R-configuration 3-substituted-3-hydroxy oxindole compound 陕西师范大学 2020-12-22 CN disclosed