SCHEMBL3467352

SCHEMBL3467352

O=C(O)c1cccc(CC2Cc3cc(-c4ccc(C(F)(F)F)cc4)ccc3NC2=O)c1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KIF11 P52732 1/20 0.45
MRGPRX4 Q96LA9 5/20 0.44
DHODH Q02127 1/20 0.40
FFAR1 O14842 1/20 0.39
TDP2 O95551 2/20 0.39
ADRB1 P08588 1/20 0.38
ADRB3 P13945 1/20 0.38
CCKAR P32238 1/20 0.38
CCKBR P32239 1/20 0.38
TDO2 P48775 1/20 0.37
NR4A2 P43354 1/20 0.37
RXRA P19793 1/20 0.37
NR1H2 P55055 1/20 0.37
NR1H3 Q13133 1/20 0.37
MEN1 O00255 1/20 0.37
KMT2A Q03164 1/20 0.37
P2RY14 Q15391 3/20 0.36
TMEM97 Q5BJF2 2/20 0.36
SIGMAR1 Q99720 2/20 0.36
KCNH2 Q12809 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3468115 0.89 KIF11 (0.47) KIF11FFAR1TDP2ADRB1ADRB3
SCHEMBL3467348 0.87 KIF11 (0.41) KIF11FFAR1
SCHEMBL3468263 0.80 KIF11 (0.53) KIF11FFAR1TDP2ADRB1ADRB3
SCHEMBL3308412 0.80 KIF11 (0.53) KIF11TDP2ADRB1ADRB3CCKAR
SCHEMBL3467503 0.80 KIF11 (0.44) KIF11FFAR1TDP2ADRB1ADRB3
SCHEMBL4891219 0.79 KIF11 (0.56) KIF11FFAR1TDP2ADRB1ADRB3
SCHEMBL3467592 0.77 KIF11 (0.52) KIF11DHODHTDP2ADRB1ADRB3
SCHEMBL4594888 0.74 KIF11 (0.56) KIF11DHODHTDP2ADRB1ADRB3
SCHEMBL3467771 0.74 KIF11 (0.48) KIF11FFAR1TDP2RXRANR1H2
SCHEMBL3467252 0.74 KIF11 (0.53) KIF11FFAR1TDP2MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010074807-A1 3, 4-DIHYDROQUINOLIN-2 ( 1H ) -ONE DERIVATIVES AS SODIUM CHANNEL MODULATORS GILEAD PALO ALTO, INC. (US) 2010-07-01 WO disclosed