SCHEMBL3469250

SCHEMBL3469250

Brc1c[nH]nc1C1CCCCO1

nearest known ligand 0.35

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
MAPK8 P45983 1/20 0.30
MAPK9 P45984 1/20 0.30
MAPK10 P53779 1/20 0.30
KCNH2 Q12809 1/20 0.30
HRH3 Q9Y5N1 1/20 0.30
PRKAB2 O43741 2/20 0.30
PRKAG1 P54619 2/20 0.30
PRKAA2 P54646 2/20 0.30
PRKAA1 Q13131 2/20 0.30
PRKAG3 Q9UGI9 2/20 0.30
PRKAG2 Q9UGJ0 2/20 0.30
PRKAB1 Q9Y478 2/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21001854 1.00 MAPK8 (0.30) MAPK8MAPK9MAPK10KCNH2HRH3
SCHEMBL26130701 0.81 PRKAB2 (0.35) PRKAB2PRKAG1PRKAA2PRKAA1PRKAG3
SCHEMBL27248736 0.80 GHSR (0.31) KCNH2HRH3
SCHEMBL17713790 0.80 PRKAG1 (0.31) KCNH2HRH3PRKAB2PRKAG1PRKAA2
SCHEMBL25293416 0.78 PLK1 (0.31)
SCHEMBL21465720 0.76
SCHEMBL28881758 0.76 ALDH1A1 (0.31)
SCHEMBL20077896 0.74 PDE5A (0.34)
SCHEMBL29218326 0.74 IRAK4 (0.35) PRKAB2PRKAG1PRKAA2PRKAA1PRKAG3
SCHEMBL21465726 0.73

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3814357-A1 HETEROCYCLIC AND HETEROARYL COMPOUNDS FOR TREATING HUNTINGTON'S DISEASE PTC Therapeutics, Inc. (US) 2021-05-05 EP disclosed
EP-2215085-A2 PYRIDINE AND PYRAZINE DERIVATIVES USEFUL IN THE TREATMENT OF CELL PROLIFERATIVE DISORDERS AstraZeneca AB (SE) 2010-08-11 EP disclosed
WO-2009053737-A2 PYRIDINE AND PYRAZINE DERIVATIVES USEFUL IN THE TREATMENT OF CELL PROLIFERATIVE DISORDERS ASTRAZENECA AB (SE) 2009-04-30 WO disclosed