SCHEMBL347122

SCHEMBL347122

O=c1ccc2cc(Br)ccc2[nH]1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 O43570 3/20 0.60
CA9 Q16790 3/20 0.60
F11 P03951 1/20 0.60
IDO1 P14902 1/20 0.54
MAPT P10636 2/20 0.52
CA1 P00915 1/20 0.52
CA3 P07451 1/20 0.52
CA4 P22748 1/20 0.52
CA6 P23280 1/20 0.52
CA5A P35218 1/20 0.52
CA7 P43166 1/20 0.52
CA13 Q8N1Q1 1/20 0.52
CA14 Q9ULX7 1/20 0.52
CA5B Q9Y2D0 1/20 0.52
CYP2A6 P11509 2/20 0.50
AHR P35869 1/20 0.50
NR4A2 P43354 1/20 0.50
AR P10275 1/20 0.47
CYP19A1 P11511 1/20 0.46
PDE3B Q13370 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL706857 0.85 CA12 (0.54) CA12CA9F11IDO1MAPT
SCHEMBL30176791 0.85 CA12 (0.54) CA12CA9F11IDO1MAPT
SCHEMBL25904886 0.85 PDE3B (0.46) CA12CA9F11IDO1MAPT
SCHEMBL5788472 0.83 F11 (0.51) CA12CA9F11IDO1MAPT
SCHEMBL6031111 0.77 CA12 (0.62) CA12CA9F11IDO1MAPT
Acetic Acid SCHEMBL9409744 0.76 HRH4 (0.47) CA12CA9F11MAPTCA1
SCHEMBL14279696 0.75 CA12 (0.60) CA12CA9F11IDO1MAPT
SCHEMBL3368797 0.75 CA12 (0.60) CA12CA9F11CA1CA3
SCHEMBL1052487 0.75 F11 (1.00) CA12CA9F11MAPTCA1
SCHEMBL5548525 0.75 AHR (0.55) MAPTCYP2A6AHRNR4A2CYP19A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 343 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20260078117-A1 COMPOUNDS AND METHODS OF USE TANGO THERAPEUTICS INC (US) 2026-03-19 US disclosed
EP-4615824-A1 SUBSTITUTED QUINOLONE COMPOUNDS USEFUL AS INHIBITORS OF TLR9 Bristol-Myers Squibb Company (US) 2025-09-17 EP disclosed
CN-120152957-A Substituted quinolones useful as TLR9 inhibitors 百时美施贵宝公司 2025-06-13 CN disclosed
EP-4561561-A2 SUBSTITUTED 3,4-DIHYDROQUINOLINONE INHIBITORS OF TSHR Septerna, Inc. (US) 2025-06-04 EP disclosed
US-12304907-B2 Compounds and methods of use TANGO THERAPEUTICS, INC. (US) 2025-05-20 US disclosed
US-20250136592-A1 C-LINKED INHIBITORS OF ENL/AF9 YEATS BRIDGE MEDICINES 2025-05-01 US disclosed
CN-115427035-B ENL/AF9 YEATS inhibitors 洛克菲勒大学 2025-04-22 CN disclosed
US-12264154-B2 Compounds and methods of use TANGO THERAPEUTICS, INC. (US) 2025-04-01 US disclosed
US-20240400499-A1 NOVEL AMINO ACID DERIVATIVES PEPTIDREAM INC (JP) 2024-12-05 US disclosed
US-20240279219-A1 COMPOUNDS AND METHODS OF USE TANGO THERAPEUTICS, INC. 2024-08-22 US disclosed
EP-0894088-A1 SUBSTITUTED SULFONIC ACID N- (AMINOIMINOMETHYL)PHENYLALKYL]-AZAHETEROCYCLAMIDE COMPOUNDS RHONE-POULENC RORER PHARMACEUTICALS, INC. (US) 1999-02-03 EP disclosed
WO-1998024784-A1 SUBSTITUTED SULFONIC ACID N-[(AMINOIMINOMETHYL)PHENYLALKYL]-AZAHETEROCYCLAMIDE COMPOUNDS RHONE-POULENC RORER PHARMACEUTICALS INC. (US) 1998-06-11 WO disclosed
US-5731315-A Substituted sulfonic acid n- (aminoiminomethyl)phenylalkyl!-azaheterocyclamide compounds RHONE-POULENC RORER PHARMACEUTICALS INC. (US) 1998-03-24 US disclosed
EP-0190857-B1 QUINOLONE INOTROPIC AGENTS Pfizer Limited (GB) 1990-03-21 EP disclosed
US-4728654-A CONGESTIVE HEART FAILURE PFIZER INC. (US) 1988-03-01 US disclosed
US-4710507-A Quinolone inotropic agents PFIZER INC. (US) 1987-12-01 US disclosed
CN-85100796-A The preparation method of qualone derivative 1986-10-01 CN disclosed
EP-0190857-A2 Quinolone inotropic agents Pfizer Limited (GB) 1986-08-13 EP disclosed
EP-0148623-A2 Quinolone inotropic agents Pfizer Limited (GB) 1985-07-17 EP disclosed
US-4236912-A Quinolinyloxyphenoxy and quinolyinylthiophenoxy alkanoic acids and derivatives thereof and methods of herbicidal use THE DOW CHEMICAL COMPANY (US) 1980-12-02 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (6 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20240279219-A1 COMPOUNDS AND METHODS OF USE F12, C1R, ABCG2 CA12 1198/4885CA9 647/4885F11 606/4885
US-12264154-B2 Compounds and methods of use F12, C1R, ABCG2 CA12 1198/4885CA9 647/4885F11 606/4885
US-12304907-B2 Compounds and methods of use F12, C1R, ABCG2 CA12 1198/4885CA9 647/4885F11 606/4885
US-20260078117-A1 COMPOUNDS AND METHODS OF USE NR3C2, ADRA1A, CNR1 CA12 522/4885CA9 339/4885F11 2491/4885
US-20250136592-A1 C-LINKED INHIBITORS OF ENL/AF9 YEATS MLLT3, MLLT1, YEATS2 CA12 4464/4885CA9 521/4885F11 3145/4885
US-20240400499-A1 NOVEL AMINO ACID DERIVATIVES BCAT1, BCAT2, PELP1 CA12 4083/4885CA9 4188/4885F11 2888/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.