SCHEMBL3474700

SCHEMBL3474700

CC(C)c1nc2c(=O)n(C3CCCCC3)c(=O)nc-2n(C2CCCCC2)n1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDP2 O95551 4/20 0.37
MEN1 O00255 3/20 0.36
KMT2A Q03164 3/20 0.36
ALDH1A1 P00352 2/20 0.36
CYP1A2 P05177 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2D6 P10635 1/20 0.36
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36
STAT3 P40763 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
GAA P10253 1/20 0.35
ALOX15 P16050 1/20 0.35
HCAR1 Q9BXC0 2/20 0.34
KDM4E B2RXH2 1/20 0.33
HSD17B10 Q99714 1/20 0.33
CRHBP P24387 1/20 0.33
CRHR2 Q13324 1/20 0.33
RXFP1 Q9HBX9 1/20 0.33
CCNT1 O60563 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3473636 0.87 TDP2 (0.48) TDP2MEN1KMT2AALDH1A1CYP1A2
SCHEMBL3474307 0.86 TDP2 (0.36) TDP2MEN1KMT2AALDH1A1CYP1A2
SCHEMBL3471025 0.73 TDP2 (0.56) TDP2MEN1KMT2AALDH1A1CYP1A2
SCHEMBL3471235 0.70 TDP2 (0.74) TDP2MEN1KMT2AALDH1A1CYP1A2
SCHEMBL3472911 0.66 TDP2 (0.37) TDP2MEN1KMT2AALDH1A1CYP1A2
SCHEMBL24610237 0.64 GPR119 (0.30)
SCHEMBL3471912 0.64 TDP2 (0.66) TDP2MEN1KMT2AALDH1A1CYP1A2
SCHEMBL18655421 0.64 ALDH1A1 (0.39) MEN1KMT2AALDH1A1CYP1A2CYP3A4
SCHEMBL24094149 0.62 CCNT1 (0.32) CCNT1CDK9
SCHEMBL3476272 0.61 TDP2 (0.40) TDP2MEN1KMT2AALDH1A1CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010072807-A2 INHIBITORS OF CYSTATHIONINE BETA SYNTHASE TO REDUCE THE NEUROTOXIC OVERPRODUCTION OF ENDOGENOUS HYDROGEN SULFIDE FONDATION JEROME LEJEUNE (FR) 2010-07-01 WO disclosed
WO-2010072807-A2 INHIBITORS OF CYSTATHIONINE BETA SYNTHASE TO REDUCE THE NEUROTOXIC OVERPRODUCTION OF ENDOGENOUS HYDROGEN SULFIDE FONDATION JEROME LEJEUNE (FR) 2010-07-01 WO disclosed