Sulfisomidine

Sulfisomidine

SCHEMBL34791

Cc1cc(NS(=O)(=O)c2ccc(N)cc2)nc(C)n1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
PDE4A P27815 1/20 1.00
AGO2 Q9UKV8 1/20 1.00
ALDH1A1 P00352 6/20 0.70
KDM4E B2RXH2 3/20 0.70
LMNA P02545 2/20 0.70
CYP3A4 P08684 3/20 0.66
SMN1; SMN2 Q16637 1/20 0.66
TDP1 Q9NUW8 1/20 0.66
HTR6 P50406 5/20 0.61
POLB P06746 3/20 0.60
MAPT P10636 3/20 0.59
CYP2C9 P11712 1/20 0.59
CYP2C19 P33261 1/20 0.59
RAB9A P51151 1/20 0.59
ADRA1A P35348 1/20 0.58
USP2 O75604 1/20 0.58
APEX1 P27695 1/20 0.58
BLM P54132 1/20 0.58
NPSR1 Q6W5P4 1/20 0.58

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Sulfisomidine SCHEMBL284793 0.98 PDE4A (0.97) PDE4AAGO2ALDH1A1KDM4ELMNA
Sulfamethazine SCHEMBL28086389 0.93 PDE4A (0.87) PDE4AAGO2ALDH1A1KDM4ELMNA
SCHEMBL1828300 0.85 PDE4A (0.74) PDE4AAGO2ALDH1A1KDM4ELMNA
SCHEMBL1381858 0.84 PDE4A (0.73) PDE4AAGO2ALDH1A1KDM4ELMNA
SCHEMBL5453637 0.83 PDE4A (0.71) PDE4AAGO2ALDH1A1KDM4ELMNA
Sulfametomidine SCHEMBL30336540 0.83 HTR6 (0.76) PDE4AAGO2ALDH1A1KDM4ELMNA
Sulfametomidine SCHEMBL151238 0.83 HTR6 (0.76) PDE4AAGO2ALDH1A1KDM4ELMNA
Sulfametomidine SCHEMBL11123046 0.82 ALDH1A1 (0.74) PDE4AAGO2ALDH1A1KDM4ELMNA
SCHEMBL11757838 0.82 PDE4A (0.69) PDE4AAGO2ALDH1A1KDM4ELMNA
SCHEMBL290584 0.80 ALDH1A1 (0.71) PDE4AAGO2ALDH1A1KDM4ELMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 4788 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20260091119-A1 ISOLATED TARGETED DELIVERY SYSTEM FOR THE TREATMENT OF GLIOMA CELLIS AG (CH) 2026-04-02 US claimed
EP-4637829-A1 ISOLATED TARGETED DELIVERY SYSTEM FOR THE TREATMENT OF OVARIAN CANCER Cellis Sp. z o.o. ([Ltd.] (PL) 2025-10-29 EP claimed
EP-4587062-A1 ISOLATED TARGETED DELIVERY SYSTEM FOR THE TREATMENT OF GLIOMA Cellis AG (CH) 2025-07-23 EP claimed
EP-4552661-A2 MEDICAL DEVICES HAVING ANTI-MICROBIAL PROPERTIES AND METHODS FOR MAKING THE SAME Hollister Incorporated (US) 2025-05-14 EP claimed
EP-4552693-A2 COLLAGEN PEPTIDE-BASED MEDICAMENT COMPOSITIONS AND DEVICES AND METHODS OF PRODUCTION AND USE THEREOF Sustain Holdings, LLC (US) 2025-05-14 EP claimed
EP-4178637-B1 MEDICAL DEVICES HAVING ANTI-MICROBIAL PROPERTIES AND METHODS FOR MAKING THE SAME HOLLISTER INC (US) 2025-05-14 EP claimed
WO-2025080590-A1 CO-CRYSTALLIZATION OF ACTIVES WITH SACCHARIDE-BASED MOLECULAR FRAMEWORKS SCIENTIFIC HORIZONS CONSULTING LLC (US) 2025-04-17 WO claimed
EP-4536217-A1 CO-AGENTS AS THERAPY AGAINST ANAEROBIC PATHOGENS Fleurir Abx LLC (US) 2025-04-16 EP claimed
US-12274830-B2 Nitric oxide inhalation therapy for infants with bronchiolitis BEYOND AIR LTD (IL) 2025-04-15 US claimed
US-20250099557-A1 ANTIBIOTIC PHARMACEUTICAL COMPOSITION CAPABLE OF SUBCUTANEOUS ADMINISTRATION SHANGHAI BAO PHARMACEUTICALS CO., LTD. (CN) 2025-03-27 US claimed
WO-1996012487-A1 COMBINATION METHOD FOR ACNE TREATMENT MERCK & CO., INC. (US) 1996-05-02 WO claimed
WO-1995020387-A1 METHOD FOR PREVENTING OR REDUCING PHOTOSENSITIVITY AND/OR PHOTOTOXICITY REACTIONS TO MEDICATIONS G.D. SEARLE & CO. (US) 1995-08-03 WO claimed
EP-0572560-A4 USE OF PHARMACEUTICAL COMPOUNDS IN THE TREATMENT OF SYMPTOMS OF DISORDERS RELATED TO NEUROLOGICAL DISEASES AND ETIOLOGICALLY RELATED SYMPTOMOLOGY. SHAPIRO HOWARD K (US) 1995-04-26 EP claimed
US-5288503-A WATER-PERMEABLE DIFFUSION BARRIER OF POLYVINYL ALCOHOL SRCHEM INCORPORATED (US) 1994-02-22 US claimed
EP-0572560-A1 USE OF PHARMACEUTICAL COMPOUNDS IN THE TREATMENT OF SYMPTOMS OF DISORDERS RELATED TO NEUROLOGICAL DISEASES AND ETIOLOGICALLY RELATED SYMPTOMOLOGY SHAPIRO, Howard, K. (US) 1993-12-08 EP claimed
US-5260066-A Cryogel bandage containing therapeutic agent SRCHEM INCORPORATED (US) 1993-11-09 US claimed
WO-1992014456-A1 USE OF PHARMACEUTICAL COMPOUNDS IN THE TREATMENT OF SYMPTOMS OF DISORDERS RELATED TO NEUROLOGICAL DISEASES AND ETIOLOGICALLY RELATED SYMPTOMOLOGY SHAPIRO HOWARD K (US) 1992-09-03 WO claimed
US-4743910-A Frequency domain, pulse compression radar apparatus for eliminating clutter HUGHES AIRCRAFT COMPANY (US) 1988-05-10 US claimed
US-4725355-A SULFA DRUG ON SUPPORT TERUMO KABUSHIKI KAISHA (JP) 1988-02-16 US claimed
US-4315931-A MICROBIOCIDES, INFECTIOUS DISEASES BASF AKTIENGESELLSCHAFT (DE) 1982-02-16 US claimed