SCHEMBL3480451

SCHEMBL3480451

O=c1ccc(-c2ccc(S(=O)(=O)NCP(=O)(O)O)s2)c[nH]1

nearest known ligand 0.46

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ATIC P31939 1/20 0.46
RORC P51449 1/20 0.36
KMT2A Q03164 2/20 0.35
POLB P06746 1/20 0.35
MEN1 O00255 1/20 0.35
PKM P14618 1/20 0.35
RAB9A P51151 1/20 0.35
MAP3K5 Q99683 2/20 0.34
MMP2 P08253 5/20 0.34
MMP9 P14780 5/20 0.34
P2RY14 Q15391 4/20 0.31
LIPC P11150 1/20 0.31
LIPG Q9Y5X9 1/20 0.31
IRAK4 Q9NWZ3 1/20 0.30
MMP13 P45452 2/20 0.30
MMP3 P08254 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3480489 0.78 SNCA (0.47) POLBP2RY14
SCHEMBL3480501 0.74 MAPT (0.48) KMT2AMEN1MMP2MMP9MMP13
SCHEMBL3480434 0.73 MMP13 (0.45) KMT2APOLBMEN1MMP2MMP9
SCHEMBL4427998 0.70 SMN1; SMN2 (0.55) KMT2AMEN1RAB9A
SCHEMBL16667405 0.70 P2RY14 (0.38) MAP3K5MMP2MMP9P2RY14MMP13
SCHEMBL3480416 0.69 MAP3K5 (0.35) KMT2APOLBMEN1PKMRAB9A
SCHEMBL3480347 0.65 MCL1 (0.41) KMT2AMEN1RAB9A
SCHEMBL3483578 0.63 L3MBTL1 (0.38) KMT2AMEN1
SCHEMBL1864479 0.63 RAB9A (0.57) KMT2APOLBMEN1RAB9A
SCHEMBL4430974 0.63 CYP2D6 (0.64) KMT2APOLBPKMRAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20100317625-A1 NOVEL SULFONAMIDOMETHYLPHOSPHONATE INHIBITORS OF BETA-LACTAMASE 92229129 QUEBEC INC. (CA) 2010-12-16 US claimed
EP-2024376-A1 NOVEL SULFONAMIDOMETHYLPHOSPHONATE INHIBITORS OF BETA-LACTAMASE Merck & Co., Inc. (US) 2009-02-18 EP claimed
WO-2007139729-A1 NOVEL SULFONAMIDOMETHYLPHOSPHONATE INHIBITORS OF BETA-LACTAMASE MERCK & CO., INC. (US) 2007-12-06 WO claimed
US-20100317625-A1 NOVEL SULFONAMIDOMETHYLPHOSPHONATE INHIBITORS OF BETA-LACTAMASE 92229129 QUEBEC INC. (CA) 2010-12-16 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100317625-A1 NOVEL SULFONAMIDOMETHYLPHOSPHONATE INHIBITORS OF BETA-LACTAMASE MGAM, BPGM, PPME1 ATIC 387/4885RORC 3260/4885KMT2A 2187/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.