Xanthine

Xanthine

SCHEMBL3514682

O=P(O)(O)O.O=P(O)(O)O.O=P(O)(O)O.O=c1[nH]c(=O)c2[nH]cnc2[nH]1

nearest known ligand 0.82

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

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

The experimentally established mechanism targets of Xanthine. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
GDA Q9Y2T3 3/20 0.82
ACHE P22303 1/20 0.82
ABL1 P00519 1/20 0.42
RIN1 Q13671 1/20 0.42
ADORA2B P29275 6/20 0.41
ADORA2A P29274 3/20 0.41
ALDH1A1 P00352 1/20 0.39
PNP P00491 1/20 0.39
PDE4A P27815 2/20 0.38
PDE4B Q07343 2/20 0.38
PDE4C Q08493 2/20 0.38
PDE4D Q08499 2/20 0.38
TDP1 Q9NUW8 1/20 0.38
ADORA3 P0DMS8 4/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Xanthine SCHEMBL389887 1.00 GDA (0.82) GDAACHEABL1RIN1ADORA2B
Xanthine SCHEMBL27830253 0.98 GDA (0.79) GDAACHEABL1RIN1ADORA2B
Xanthine SCHEMBL4965 0.91 GDA (1.00) GDAACHEABL1RIN1ADORA2B
Xanthine SCHEMBL2352524 0.91 GDA (1.00) GDAACHEABL1RIN1ADORA2B
Xanthine SCHEMBL29669592 0.91 GDA (1.00) GDAACHEABL1RIN1ADORA2B
Xanthine SCHEMBL7849418 0.89 GDA (0.96) GDAACHEABL1RIN1ADORA2B
Xanthine SCHEMBL1507586 0.89 GDA (0.96) GDAACHEABL1RIN1ADORA2B
Xanthine SCHEMBL31488667 0.89 GDA (0.96) GDAACHEABL1RIN1ADORA2B
Xanthine SCHEMBL6783299 0.89 GDA (0.96) GDAACHEABL1RIN1ADORA2B
Xanthine SCHEMBL2454001 0.89 GDA (0.96) GDAACHEABL1RIN1ADORA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20100317005-A1 Modified Nucleotides and Methods for Making and Use Same Life Technologies Corporation (US) 2010-12-16 US claimed