Xanthine

Xanthine

SCHEMBL389887

O=P(O)(O)O.O=c1[nH]c(=O)c2[nH]cnc2[nH]1

nearest known ligand 0.82

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

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

The experimentally established mechanism targets of Xanthine. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
GDA Q9Y2T3 3/20 0.82
ACHE P22303 1/20 0.82
ABL1 P00519 1/20 0.42
RIN1 Q13671 1/20 0.42
ADORA2B P29275 6/20 0.41
ADORA2A P29274 3/20 0.41
ALDH1A1 P00352 1/20 0.39
PNP P00491 1/20 0.39
PDE4A P27815 2/20 0.38
PDE4B Q07343 2/20 0.38
PDE4C Q08493 2/20 0.38
PDE4D Q08499 2/20 0.38
TDP1 Q9NUW8 1/20 0.38
ADORA3 P0DMS8 4/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Xanthine SCHEMBL3514682 1.00 GDA (0.82) GDAACHEABL1RIN1ADORA2B
Xanthine SCHEMBL27830253 0.98 GDA (0.79) GDAACHEABL1RIN1ADORA2B
Xanthine SCHEMBL4965 0.91 GDA (1.00) GDAACHEABL1RIN1ADORA2B
Xanthine SCHEMBL2352524 0.91 GDA (1.00) GDAACHEABL1RIN1ADORA2B
Xanthine SCHEMBL29669592 0.91 GDA (1.00) GDAACHEABL1RIN1ADORA2B
Xanthine SCHEMBL7849418 0.89 GDA (0.96) GDAACHEABL1RIN1ADORA2B
Xanthine SCHEMBL1507586 0.89 GDA (0.96) GDAACHEABL1RIN1ADORA2B
Xanthine SCHEMBL31488667 0.89 GDA (0.96) GDAACHEABL1RIN1ADORA2B
Xanthine SCHEMBL6783299 0.89 GDA (0.96) GDAACHEABL1RIN1ADORA2B
Xanthine SCHEMBL2454001 0.89 GDA (0.96) GDAACHEABL1RIN1ADORA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 359 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20220218731-A1 COMBINATION THERAPIES FOR CANCER TREATMENT CLEAR CREEK BIO INC (US) 2022-07-14 US claimed
WO-2020236502-A1 COMBINATION THERAPIES FOR CANCER TREATMENT Clear Creek Bio, Inc. (US) 2020-11-26 WO claimed
US-20260116994-A1 RECOMBINANT MONOCLONAL ANTIBODIES AND CORRESPONDING ANTIGENS FOR COLON AND PANCREATIC CANCERS PREC BIOLOGICS INC (US) 2026-04-30 US disclosed
US-12584099-B2 Method for preparing cultures of lactic acid bacteria CHR. HANSEN A/S (DK) 2026-03-24 US disclosed
US-20260015432-A1 RECOMBINANT MONOCLONAL ANTIBODIES AND CORRESPONDING ANTIGENS FOR COLON AND PANCREATIC CANCERS PREC BIOLOGICS INC (US) 2026-01-15 US disclosed
US-12460013-B2 Recombinant monoclonal antibodies and corresponding antigens for colon and pancreatic cancers PRECISION BIOLOGICS, INC. (US) 2025-11-04 US disclosed
US-12344676-B2 Recombinant monoclonal antibodies and corresponding antigens for colon and pancreatic cancers PRECISION BIOLOGICS, INC. (US) 2025-07-01 US disclosed
WO-2025105871-A1 GENE EDITING TREATMENT METHOD AND THERAPEUTIC AGENT FOR RETINITIS PIGMENTOSA 재단법인 아산사회복지재단 2025-05-22 WO disclosed
US-20250049753-A1 METHODS AND COMPOSITIONS FOR DELIVERING MYCOPHENOLIC ACID ACTIVE AGENTS TO NON-HUMAN MAMMALS OKAVA PHARMACEUTICALS INC (US) 2025-02-13 US disclosed
US-20240368532-A1 METHOD FOR PREPARING CULTURES OF LACTIC ACID BACTERIA CHR. HANSEN A/S (DK) 2024-11-07 US disclosed
US-20240343825-A1 RECOMBINANT MONOCLONAL ANTIBODIES AND CORRESPONDING ANTIGENS FOR COLON AND PANCREATIC CANCERS PREC BIOLOGICS INC (US) 2024-10-17 US disclosed
WO-1989011538-A1 PLATELET-SPECIFIC CHIMERIC IMMUNOGLOBULIN CENTOCOR, INC. (US) 1989-11-30 WO disclosed
WO-1989008716-A1 NOVEL RECOMBINANT VACCINIA VIRUS EXPRESSION VECTORS AND METHOD OF SELECTING SAME THE UNITED STATES OF AMERICA, AS REPRESENTED BY TH (US) 1989-09-21 WO disclosed
EP-0322417-A1 EMPTY VIRAL CAPSID VACCINES APPLIED BIOTECHNOLOGY, INC. (US) 1989-07-05 EP disclosed
WO-1989004872-A1 IMMUNOREACTIVE HETEROCHAIN ANTIBODIES CENTOCOR, INC. (US) 1989-06-01 WO disclosed
WO-1988009181-A2 MONOCLONAL ANTIBODIES NEUTRALIZING HIV-1 TANOX BIOSYSTEMS, INC. (US) 1988-12-01 WO disclosed
WO-1988002026-A1 EMPTY VIRAL CAPSID VACCINES APPLIED BIOTECHNOLOGY, INC. (US) 1988-03-24 WO disclosed
WO-1988002022-A1 RECOMBINANT POXVIRUSES COMMONWEALTH SCIENTIFIC AND INDUSTRIAL RESEARCH OR (AU) 1988-03-24 WO disclosed
EP-0256654-A2 Chimeric murine/human immunoglobulin specific for tumour-associated 17-1A Antigen CENTOCOR, INC. (US) 1988-02-24 EP disclosed
US-4550186-A ANTITUMOR, ANTILIPEMIC, ANTIINFLAMMATORY, AND ANTIARTHRITIC AGENTS DUKE UNIVERSITY (US) 1985-10-29 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20260116994-A1 RECOMBINANT MONOCLONAL ANTIBODIES AND CORRESPONDING ANTIGENS FOR COLON AND PANCREATIC CANCERS IGSF11, IGLV6-57, VSIG8 GDA 1840/4885ACHE 4740/4885ABL1 3101/4885
US-20250049753-A1 METHODS AND COMPOSITIONS FOR DELIVERING MYCOPHENOLIC ACID ACTIVE AGENTS TO NON-HUMAN MAMMALS CD47, TPMT, HLA-C GDA 607/4885ACHE 4461/4885ABL1 1667/4885
US-20260015432-A1 RECOMBINANT MONOCLONAL ANTIBODIES AND CORRESPONDING ANTIGENS FOR COLON AND PANCREATIC CANCERS VIP, IAPP, RNASE1 GDA 467/4885ACHE 4109/4885ABL1 3299/4885
US-12584099-B2 Method for preparing cultures of lactic acid bacteria LCT, S100A10, RPLP0 GDA 1191/4885ACHE 4531/4885ABL1 3909/4885
US-20220218731-A1 COMBINATION THERAPIES FOR CANCER TREATMENT PCK2, PC, FOLR2 GDA 1214/4885ACHE 4803/4885ABL1 1416/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.