4'-Thiothymidine

4'-Thiothymidine

SCHEMBL3517588

Cc1cn([C@@H]2C[C@H](O)[C@H](CO)S2)c(=O)[nH]c1=O

nearest known ligand 0.54

Full drug profile on Sugi Atlas →

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
TK1 P04183 5/20 0.49
ALDH1A1 P00352 1/20 0.49
LMNA P02545 1/20 0.49
ALB P02768 1/20 0.49
POLB P06746 1/20 0.49
ADRA1A P35348 1/20 0.49
BLM P54132 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
4'-Thiothymidine SCHEMBL6266871 1.00 TK1 (0.49) TK1ALDH1A1LMNAALBPOLB
4'-Thiothymidine SCHEMBL1942500 1.00 TK1 (0.49) TK1ALDH1A1LMNAALBPOLB
4'-Thiothymidine SCHEMBL3517583 1.00 TK1 (0.49) TK1ALDH1A1LMNAALBPOLB
4'-Thiothymidine SCHEMBL13083838 1.00 TK1 (0.49) TK1ALDH1A1LMNAALBPOLB
4'-Thiothymidine SCHEMBL23897578 1.00 TK1 (0.49) TK1ALDH1A1LMNAALBPOLB
4'-Thiothymidine SCHEMBL6311407 1.00 TK1 (0.49) TK1ALDH1A1LMNAALBPOLB
4'-Thiothymidine SCHEMBL23897630 1.00 TK1 (0.49) TK1ALDH1A1LMNAALBPOLB
4'-Thiothymidine SCHEMBL9520953 1.00 TK1 (0.49) TK1ALDH1A1LMNAALBPOLB
4'-Thiothymidine SCHEMBL12642446 1.00 TK1 (0.49) TK1ALDH1A1LMNAALBPOLB
4'-Thiothymidine SCHEMBL30381070 1.00 TK1 (0.49) TK1ALDH1A1LMNAALBPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 22 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5591722-A ANTICANCER AGENTS SOUTHERN RESEARCH INSTITUTE (US) 1997-01-07 US claimed
EP-0491793-A4 2'-DEOXY-4'-THIORIBONUCLEOSIDES AS ANTIVIRAL AND ANTICANCER AGENTS 1993-03-03 EP claimed
EP-0491793-A1 2'-DEOXY-4'-THIORIBONUCLEOSIDES AS ANTIVIRAL AND ANTICANCER AGENTS SOUTHERN RESEARCH INSTITUTE (US) 1992-07-01 EP claimed
WO-1991004033-A1 2'-DEOXY-4'-THIORIBONUCLEOSIDES AS ANTIVIRAL AND ANTICANCER AGENTS SOUTHERN RESEARCH INSTITUTE (US) 1991-04-04 WO claimed
US-20120225837-A1 MEDICINAL AGENT FOR DISEASE ASSOCIATED WITH EPSTEIN-BARR VIRUS, AND METHOD FOR SCREENING OF THE MEDICINAL AGENT KYOTO UNIVERSITY (JP) 2012-09-06 US disclosed
EP-2189161-B1 MEDICINAL AGENT FOR DISEASE ASSOCIATED WITH EPSTEIN-BARR VIRUS, AND METHOD FOR SCREENING OF THE MEDICINAL AGENT YAMASA CORP (JP) 2012-08-08 EP disclosed
US-20100330563-A1 MEDICINAL AGENT FOR DISEASE ASSOCIATED WITH EPSTEIN-BARR VIRUS, AND METHOD FOR SCREENING OF THE MEDICINAL AGENT YAMASA CORPORATION (JP) 2010-12-30 US disclosed
EP-2189161-A1 MEDICINAL AGENT FOR DISEASE ASSOCIATED WITH EPSTEIN-BARR VIRUS, AND METHOD FOR SCREENING OF THE MEDICINAL AGENT YAMASA CORPORATION (JP) 2010-05-26 EP disclosed
EP-0491793-B1 2'-DEOXY-4'-THIORIBONUCLEOSIDES AS ANTIVIRAL AND ANTICANCER AGENTS SOUTHERN RES INST (US) 2005-11-30 EP disclosed
US-6949522-B2 β-2′- or 3′-halonucleosides PHARMASSET, INC. (US) 2005-09-27 US disclosed
US-20050119286-A1 BETA-2'-OR 3'-HALONUCLEOSIDES NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2005-06-02 US disclosed
EP-1478322-A2 Beta-2'-OR 3'-HALONUCLEOSIDES Pharmasset Limited (BB) 2004-11-24 EP disclosed
US-5478928-A Useful as antiviral agents in the treatment and prevention of AIDS SOUTHERN RESEARCH INSTITUTE (US) 1995-12-26 US disclosed
EP-0525106-A4 2',3'-DIDEOXY-4'-THIORIBONUCLEOSIDES AS ANTIVIRAL AGENTS 1993-04-21 EP disclosed
EP-0491793-A4 2'-DEOXY-4'-THIORIBONUCLEOSIDES AS ANTIVIRAL AND ANTICANCER AGENTS 1993-03-03 EP disclosed
EP-0525106-A1 2',3'-DIDEOXY-4'-THIORIBONUCLEOSIDES AS ANTIVIRAL AGENTS SOUTHERN RESEARCH INSTITUTE (US) 1993-02-03 EP disclosed
US-5128458-A 2',3'-dideoxy-4'-thioribonucleosides as antiviral agents SOUTHERN RESEARCH INSTITUTE (US) 1992-07-07 US disclosed
EP-0491793-A1 2'-DEOXY-4'-THIORIBONUCLEOSIDES AS ANTIVIRAL AND ANTICANCER AGENTS SOUTHERN RESEARCH INSTITUTE (US) 1992-07-01 EP disclosed
WO-1991016333-A1 2',3'-DIDEOXY-4'-THIORIBONUCLEOSIDES AS ANTIVIRAL AGENTS SOUTHERN RESEARCH INSTITUTE (US) 1991-10-31 WO disclosed
WO-1991004033-A1 2'-DEOXY-4'-THIORIBONUCLEOSIDES AS ANTIVIRAL AND ANTICANCER AGENTS SOUTHERN RESEARCH INSTITUTE (US) 1991-04-04 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050119286-A1 BETA-2'-OR 3'-HALONUCLEOSIDES MKI67, EBP, PCNA TK1 157/4885ALDH1A1 2973/4885LMNA 211/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.