SCHEMBL3521701

SCHEMBL3521701

Cc1ccccc1Nc1ccc(Cl)cc1NC=O

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 3/20 0.42
ALDH1A1 P00352 5/20 0.41
MAPT P10636 3/20 0.41
TP53 P04637 1/20 0.41
RAPGEF4 Q8WZA2 1/20 0.41
KCNMA1 Q12791 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.38
MAPK13 O15264 1/20 0.38
MAPK12 P53778 1/20 0.38
MAPK11 Q15759 1/20 0.38
MAPK14 Q16539 1/20 0.38
KDM4E B2RXH2 2/20 0.38
MEN1 O00255 1/20 0.38
HSP90AA1 P07900 1/20 0.38
HSP90AB1 P08238 1/20 0.38
GAA P10253 1/20 0.38
THRB P10828 1/20 0.38
HPGD P15428 1/20 0.38
BLM P54132 1/20 0.38
KMT2A Q03164 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1758540 0.80 RAPGEF4 (0.50) LMNAALDH1A1MAPTRAPGEF4KDM4E
SCHEMBL7529692 0.77 MAPK1 (0.50) ALDH1A1MAPTTP53RAPGEF4SMN1; SMN2
SCHEMBL11412614 0.77 MAPK1 (0.50) ALDH1A1MAPTTP53RAPGEF4SMN1; SMN2
SCHEMBL225741 0.76 NPC1 (0.50) ALDH1A1MAPTKDM4EGAAHPGD
SCHEMBL9800976 0.76 NPC1 (0.50) ALDH1A1MAPTKDM4EGAAHPGD
SCHEMBL14514318 0.74 CXCR2 (0.52) LMNAALDH1A1MAPTRAPGEF4KCNMA1
SCHEMBL11409022 0.74 NPC1 (0.48) ALDH1A1MAPTKDM4EGAAHPGD
SCHEMBL22313979 0.74 ALDH1A1 (0.42) LMNAALDH1A1MAPTRAPGEF4KCNMA1
SCHEMBL1713041 0.72 HTT (0.56) LMNAALDH1A1MAPTTP53SMN1; SMN2
SCHEMBL2329868 0.72 L3MBTL1 (0.51) LMNAALDH1A1MAPTSMN1; SMN2MAPK13

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7737136-B2 Non-steroidal progesterone receptor modulators N.V. ORGANON (NL) 2010-06-15 US disclosed
EP-1495030-B1 NON-STEROIDAL PROGESTERONE RECEPTOR MODULATORS ORGANON NV (NL) 2008-08-13 EP disclosed
US-20050171087-A1 Non-steroidal progesterone receptor modulators MERCK SHARP & DOHME B.V. (NL) 2005-08-04 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050171087-A1 Non-steroidal progesterone receptor modulators PGR, PGRMC1, PGRMC2 LMNA 4247/4885ALDH1A1 1163/4885MAPT 4359/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.