SCHEMBL3524858

SCHEMBL3524858

Cc1ccccc1-c1cc(NC(=O)C(C)C)cc2c1CCN(C(=O)C(F)(F)F)C2

nearest known ligand 0.42

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
PDK2 Q15119 1/20 0.42
ESR1 P03372 3/20 0.39
ESR2 Q92731 3/20 0.39
ABHD6 Q9BV23 1/20 0.39
CREBBP Q92793 4/20 0.38
EP300 Q09472 1/20 0.38
BTK Q06187 1/20 0.38
NPC1 O15118 3/20 0.38
RAB9A P51151 3/20 0.38
KMT2A Q03164 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.36
THRB P10828 1/20 0.36
NPY5R Q15761 1/20 0.35
MLYCD O95822 1/20 0.35
NAMPT P43490 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL169273 0.90 PDK2 (0.41) PDK2ESR1ESR2ABHD6CREBBP
SCHEMBL3528315 0.89 NOTUM (0.43) PDK2CREBBPEP300NPC1RAB9A
SCHEMBL3527784 0.85 CDK4 (0.44) NPC1RAB9ASMN1; SMN2NAMPT
SCHEMBL3529114 0.83 ESR1 (0.44) ESR1ESR2ABHD6CREBBPEP300
SCHEMBL169287 0.78 NOTUM (0.42) PDK2NPC1RAB9AKMT2ASMN1; SMN2
SCHEMBL16104413 0.76 RAB9A (0.42) PDK2NPC1RAB9AKMT2ASMN1; SMN2
SCHEMBL2129261 0.75 ITGB2 (0.42) SMN1; SMN2NAMPT
SCHEMBL3533607 0.74 KMT2A (0.42) PDK2NPC1RAB9AKMT2ASMN1; SMN2
SCHEMBL13076550 0.74 TMPRSS2 (0.46) ESR1ESR2NPC1RAB9AKMT2A
SCHEMBL3434989 0.73 NAMPT (0.45) ESR1ESR2NPC1RAB9AKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20120101115-A1 Compounds For Inducing Cellular Apoptosis QUEEN MARY AND WESTFIELD COLLEGE (GB) 2012-04-26 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120101115-A1 Compounds For Inducing Cellular Apoptosis BAD, BAX, CASP3 PDK2 437/4885ESR1 3474/4885ESR2 2946/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.