SCHEMBL3525912

SCHEMBL3525912

O=C(O)c1c(F)ccc2nn[nH]c12

nearest known ligand 0.33

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
HAO1 Q9UJM8 5/20 0.33
IDO1 P14902 1/20 0.33
TDO2 P48775 1/20 0.33
HCAR2 Q8TDS4 1/20 0.32
CA12 O43570 1/20 0.32
ALPL P05186 1/20 0.32
RPA1 P27694 1/20 0.32
DHODH Q02127 2/20 0.31
CES2 O00748 1/20 0.31
CES1 P23141 1/20 0.31
ALDH1A1 P00352 1/20 0.31
CAT P04040 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3522910 0.77 PDE4D (0.42) CA12ALPLALDH1A1
SCHEMBL30798651 0.72 PARP1 (0.37) ALDH1A1
SCHEMBL18226070 0.72 PARP1 (0.37) ALDH1A1
SCHEMBL17084662 0.72 TSHR (0.39) ALPLALDH1A1
SCHEMBL18528856 0.70 MAPK1 (0.36) HAO1HCAR2CA12ALPLRPA1
SCHEMBL3309453 0.70 CES2 (0.50) CA12CES2CES1ALDH1A1CAT
SCHEMBL21120441 0.70
SCHEMBL30048528 0.70 CES2 (0.50) CA12CES2CES1ALDH1A1CAT
SCHEMBL2426508 0.69 CYP19A1 (0.36) HAO1HCAR2ALDH1A1
SCHEMBL24949698 0.69 KDM4E (0.38) HCAR2ALPLDHODHALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7645771-B2 CCR5 antagonists as therapeutic agents SMITHKLINE BEECHAM CORP. (US) 2010-01-12 US disclosed
US-7645771-B2 CCR5 antagonists as therapeutic agents SMITHKLINE BEECHAM CORP. (US) 2010-01-12 US disclosed
US-7645771-B2 CCR5 antagonists as therapeutic agents SMITHKLINE BEECHAM CORP. (US) 2010-01-12 US disclosed
US-20060229336-A1 Ccr5 antagonists as therapeutic agents SMITHKLINE BEECHAM CORPORATION 2006-10-12 US disclosed
CN-1744899-A Piperidine derivatives as CCR5 antagonists SMITHKLINE BEECHAM CORP (US) 2006-03-08 CN disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060229336-A1 Ccr5 antagonists as therapeutic agents CCR5, CCR1, CXCR3 HAO1 2982/4885IDO1 108/4885TDO2 2866/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.