SCHEMBL3530225

SCHEMBL3530225

CCOC(=O)c1cn(Cc2ccccc2)c2nc(S(=O)(=O)CC)ncc2c1=O

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.51
MAPK1 P28482 1/20 0.51
ALDH1A1 P00352 3/20 0.47
KDM4E B2RXH2 2/20 0.47
P2RX3 P56373 1/20 0.46
RAB9A P51151 2/20 0.46
MEN1 O00255 1/20 0.46
NPC1 O15118 1/20 0.46
LMNA P02545 1/20 0.46
HPGD P15428 1/20 0.46
HTT P42858 1/20 0.46
KMT2A Q03164 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.46
P2RX7 Q99572 1/20 0.46
TDP1 Q9NUW8 1/20 0.45
CRHBP P24387 1/20 0.44
CRHR2 Q13324 1/20 0.44
MAPT P10636 2/20 0.42
CSF1R P07333 1/20 0.42
NPSR1 Q6W5P4 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3533125 0.92 MAPK1 (0.51) TSHRMAPK1ALDH1A1KDM4EP2RX3
SCHEMBL3526298 0.83 TSHR (0.54) TSHRMAPK1ALDH1A1KDM4EP2RX3
SCHEMBL11873809 0.79 LMNA (0.52) TSHRMAPK1ALDH1A1KDM4EMEN1
SCHEMBL3293573 0.77 CSF1R (0.44) TSHRMAPK1ALDH1A1KDM4ERAB9A
SCHEMBL11583159 0.75 LMNA (0.59) TSHRMAPK1ALDH1A1KDM4EMEN1
SCHEMBL15956289 0.74 LMNA (0.70) ALDH1A1P2RX3LMNATP53F2RL3
SCHEMBL3529229 0.74 CSF1R (0.79) CSF1R
SCHEMBL3533106 0.73 CSF1R (0.65) CSF1R
SCHEMBL11582004 0.73 ALDH1A1 (0.53) TSHRMAPK1ALDH1A1KDM4ERAB9A
SCHEMBL4574269 0.72 CSF1R (0.46) TSHRMAPK1ALDH1A1KDM4ERAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7642270-B2 5-oxo-5,8-dihydro-pyrido-pyrimidine as inhibitors of c-fms kinase JANSSEN PHARMACEUTICA N.V. (BE) 2010-01-05 US disclosed
US-20070060577-A1 5-Oxo-5,8-dihydro-pyrido-pyrimidines as inhibitors of c-fms kinase JANSSEN PHARMACEUTICA N.V. (BE) 2007-03-15 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070060577-A1 5-Oxo-5,8-dihydro-pyrido-pyrimidines as inhibitors of c-fms kinase FLT3, FES, FGR TSHR 1862/4885MAPK1 354/4885ALDH1A1 3590/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.