SCHEMBL3545167

SCHEMBL3545167

O=C(NCc1ccc(S(=O)(=O)NCC2CCCN(Cc3ccc(C(F)(F)F)cc3)C2)s1)c1ccccc1

nearest known ligand 0.50

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.50
BCHE P06276 1/20 0.46
ACKR3 P25106 1/20 0.45
MEN1 O00255 4/20 0.45
KMT2A Q03164 4/20 0.45
POLB P06746 4/20 0.45
CHRM4 P08173 1/20 0.44
CCR2 P41597 3/20 0.44
DRD2 P14416 1/20 0.43
DRD4 P21917 1/20 0.43
OPRM1 P35372 1/20 0.43
OPRK1 P41145 1/20 0.43
DDR1 Q08345 2/20 0.43
NPC1 O15118 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3547611 0.93 ALDH1A1 (0.49) ALDH1A1MEN1KMT2ACCR2DDR1
SCHEMBL3545170 0.82 POLB (0.41) ALDH1A1ACKR3MEN1KMT2APOLB
SCHEMBL3545198 0.80 CCR2 (0.54) KMT2ACCR2DDR1NPC1
SCHEMBL3544308 0.79 CCR2 (0.53) CCR2DDR1
SCHEMBL3480186 0.75 MAPK9 (0.49) ALDH1A1MEN1KMT2APOLB
SCHEMBL3546787 0.75 CCR2 (0.48) CHRM4CCR2DRD4
SCHEMBL6753597 0.74 CCR2 (0.52) MEN1KMT2ACCR2
SCHEMBL12334073 0.73 CCKBR (0.49) MEN1KMT2ANPC1
SCHEMBL3479914 0.72 MAPK9 (0.53) ALDH1A1MEN1KMT2APOLBCCR2
SCHEMBL3479910 0.72 MAPK9 (0.53) ALDH1A1MEN1KMT2APOLBCCR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7683078-B2 Arylsulfonamide derivatives as C-Jun-N-Terminal Kinases (JNK's) inhibitors LABORATOIRES SERONO S.A. (CH) 2010-03-23 US claimed