SCHEMBL3545170

SCHEMBL3545170

NC(=O)c1ccccc1Cc1ccc(S(=O)(=O)NCC2CCCN(Cc3ccc(C(F)(F)F)cc3)C2)s1

nearest known ligand 0.41

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
POLB P06746 5/20 0.41
ALDH1A1 P00352 4/20 0.41
MEN1 O00255 3/20 0.41
KMT2A Q03164 3/20 0.41
DRD4 P21917 2/20 0.39
PARP1 P09874 1/20 0.38
PARP2 Q9UGN5 1/20 0.38
ACKR3 P25106 1/20 0.38
SIGMAR1 Q99720 2/20 0.38
NPC1 O15118 1/20 0.38
LMNA P02545 1/20 0.38
MAPT P10636 1/20 0.37
KDM4E B2RXH2 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
F10 P00742 2/20 0.37
DRD2 P14416 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3545167 0.82 ALDH1A1 (0.50) POLBALDH1A1MEN1KMT2ADRD4
SCHEMBL3547611 0.79 ALDH1A1 (0.49) ALDH1A1MEN1KMT2A
SCHEMBL6753593 0.75 CCR2 (0.40) ALDH1A1KDM4ESMN1; SMN2
SCHEMBL6753601 0.73 SCN9A (0.38) ALDH1A1PARP1PARP2KDM4ESMN1; SMN2
SCHEMBL3545198 0.66 CCR2 (0.54) KMT2ANPC1
SCHEMBL3544748 0.66 SLC6A5 (0.37) ALDH1A1KMT2ASIGMAR1KDM4ESMN1; SMN2
SCHEMBL3782330 0.65 ALDH1A1 (0.59) POLBALDH1A1LMNAMAPTKDM4E
SCHEMBL13059810 0.65 ALDH1A1 (0.59) POLBALDH1A1LMNAMAPTKDM4E
SCHEMBL8328663 0.65 CYP2D6 (0.65) POLBALDH1A1LMNAMAPTKDM4E
SCHEMBL4425790 0.65 KDM4E (0.53) ALDH1A1PARP1KDM4ESMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7683078-B2 Arylsulfonamide derivatives as C-Jun-N-Terminal Kinases (JNK's) inhibitors LABORATOIRES SERONO S.A. (CH) 2010-03-23 US claimed