SCHEMBL3553263

SCHEMBL3553263

CCC(C)C(=O)NCc1sc(-c2ccc(Cl)cc2Cl)c(-c2ccc(Cl)cc2)c1C

nearest known ligand 0.37

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.37
KDM4E B2RXH2 2/20 0.37
RAB9A P51151 1/20 0.37
SHMT1 P34896 1/20 0.36
SHMT2 P34897 1/20 0.36
TP53 P04637 1/20 0.36
MDM2 Q00987 1/20 0.36
CNR1 P21554 6/20 0.36
SMN1; SMN2 Q16637 2/20 0.35
MAPT P10636 3/20 0.35
LMNA P02545 1/20 0.35
CNR2 P34972 2/20 0.35
MEN1 O00255 1/20 0.35
HPGD P15428 1/20 0.35
HTT P42858 1/20 0.35
KMT2A Q03164 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3547208 0.91 ALDH1A1 (0.40) ALDH1A1TP53MDM2CNR1CNR2
SCHEMBL3555703 0.85 ALDH1A1 (0.38) ALDH1A1TP53MDM2CNR1MAPT
SCHEMBL3550101 0.85 MMP2 (0.35) SHMT1SHMT2TP53MDM2CNR1
SCHEMBL3551713 0.83 CNR1 (0.39) ALDH1A1KDM4ECNR1SMN1; SMN2MAPT
SCHEMBL3548754 0.82 CNR1 (0.40) SHMT1SHMT2TP53MDM2CNR1
SCHEMBL3546576 0.80 P2RX7 (0.37) SHMT1SHMT2TP53CNR1MAPT
SCHEMBL3550717 0.75 MAPT (0.44) TP53MDM2CNR1MAPTLMNA
SCHEMBL5328457 0.74 HSD11B1 (0.43) ALDH1A1KDM4ERAB9ALMNAHPGD
SCHEMBL3549630 0.74 HSD11B1 (0.35) SHMT1SHMT2TP53MDM2CNR1
SCHEMBL3552068 0.74 CNR1 (0.41) TP53MDM2CNR1CNR2HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7674821-B2 N-[(4,5-diphenyl-3-alkyl-2-thienyl)methyl]amine [amide, sulfonamide, carbamate and urea) derivatives as cannabinoid CB1 receptor antagonists SANOFI-AVENTIS (FR) 2010-03-09 US claimed