SCHEMBL3566770

SCHEMBL3566770

CC(NC(CNCc1ccccc1)CC1=COCO1)c1csc(-n2ccnc2)n1

nearest known ligand 0.32

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ADRB2 P07550 1/20 0.32
ADRB1 P08588 1/20 0.32
ADRB3 P13945 1/20 0.32
PDE5A O76074 2/20 0.31
PTGS1 P23219 1/20 0.31
TBXAS1 P24557 1/20 0.31
PTGS2 P35354 1/20 0.31
PDE3B Q13370 1/20 0.31
PDE3A Q14432 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3559827 0.84 NOS2 (0.44) PDE5APTGS1TBXAS1PTGS2PDE3B
SCHEMBL3559005 0.82 NOS2 (0.38) PDE5APTGS1TBXAS1PTGS2PDE3B
SCHEMBL3563614 0.70 NOS2 (0.51) PDE5A
SCHEMBL3561919 0.69 NOS2 (0.54) PDE5A
SCHEMBL3559740 0.68 NOS2 (0.46)
SCHEMBL3571989 0.68 NOS2 (0.53) PDE5A
SCHEMBL3566764 0.67 NOS2 (0.53)
SCHEMBL3560293 0.67 NOS2 (0.48)
Hydrochloric Acid SCHEMBL3563512 0.66 NOS2 (0.48)
SCHEMBL3556543 0.66 NOS2 (0.51)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7825256-B2 Inducible nitric oxide synthase dimerization inhibitors KALYPSYS, INC. (US) 2010-11-02 US disclosed
US-20060116515-A1 Inducible nitric oxide synthase dimerization inhibitors KALYPSYS, INC. 2006-06-01 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060116515-A1 Inducible nitric oxide synthase dimerization inhibitors NOS3, NOS2, NOS1 ADRB2 1587/4885ADRB1 1018/4885ADRB3 1292/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.