SCHEMBL3561919

SCHEMBL3561919

Cc1cc(C(C)NC(CCN(C)Cc2ccccc2)CC2=COCO2)nc(-n2ccnc2)n1

nearest known ligand 0.54

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
NOS2 P35228 13/20 0.54
NOS1 P29475 2/20 0.54
HTR1D P28221 1/20 0.33
CYP1A2 P05177 2/20 0.32
CYP3A4 P08684 2/20 0.32
CYP2D6 P10635 2/20 0.32
CYP2C9 P11712 2/20 0.32
CYP2C19 P33261 2/20 0.32
ALOX15 P16050 1/20 0.32
TSHR P16473 3/20 0.32
MAPK1 P28482 2/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
NPC1 O15118 1/20 0.31
HSD17B10 Q99714 1/20 0.31
PDE5A O76074 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3563614 0.92 NOS2 (0.51) NOS2NOS1HTR1DCYP1A2CYP3A4
SCHEMBL3559827 0.85 NOS2 (0.44) NOS2NOS1PDE5A
SCHEMBL3571989 0.81 NOS2 (0.53) NOS2NOS1TSHRMAPK1NPC1
SCHEMBL3569171 0.74 NOS2 (0.41) NOS2NOS1CYP1A2CYP3A4CYP2D6
SCHEMBL3569290 0.71 NOS2 (0.57) NOS2NOS1TSHRNPC1HSD17B10
SCHEMBL3560293 0.71 NOS2 (0.48) NOS2NOS1
Hydrochloric Acid SCHEMBL3563512 0.70 NOS2 (0.48) NOS2NOS1
SCHEMBL3563611 0.70 NOS2 (1.00) NOS2NOS1
SCHEMBL3566770 0.69 ADRB2 (0.32) PDE5A
SCHEMBL3559005 0.69 NOS2 (0.38) NOS2NOS1TSHRNPC1HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7825256-B2 Inducible nitric oxide synthase dimerization inhibitors KALYPSYS, INC. (US) 2010-11-02 US disclosed
US-20060116515-A1 Inducible nitric oxide synthase dimerization inhibitors KALYPSYS, INC. 2006-06-01 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060116515-A1 Inducible nitric oxide synthase dimerization inhibitors NOS3, NOS2, NOS1 NOS2 2/4885NOS1 3/4885HTR1D 2149/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.