SCHEMBL3574238

SCHEMBL3574238

CNc1ncc(Cl)cc1C(=O)N(CCc1ccc(Cl)c(Cl)c1)Cc1ccc(C(F)(C(F)(F)F)C(F)(F)F)cc1

nearest known ligand 0.37

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
MLYCD O95822 1/20 0.35
SIGMAR1 Q99720 2/20 0.34
HSP90AA1 P07900 2/20 0.34
TRPM8 Q7Z2W7 1/20 0.34
OPRM1 P35372 1/20 0.33
OPRD1 P41143 1/20 0.33
C5AR1 P21730 1/20 0.33
CETP P11597 1/20 0.33
RAF1 P04049 1/20 0.33
MAP2K1 Q02750 1/20 0.33
TRPV1 Q8NER1 1/20 0.33
KCNH2 Q12809 2/20 0.32
TMEM97 Q5BJF2 2/20 0.32
F10 P00742 2/20 0.32
CENPE Q02224 1/20 0.32
CYP2C19 P33261 1/20 0.32
KLKB1 P03952 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3584062 0.92 GBA1 (0.34) MLYCDSIGMAR1HSP90AA1OPRM1OPRD1
SCHEMBL3569329 0.92 C5AR1 (0.41) MLYCDC5AR1F10KLKB1
SCHEMBL3576692 0.91 ESRRG (0.37) SIGMAR1HSP90AA1TRPM8OPRM1OPRD1
SCHEMBL3579477 0.90 MCHR1 (0.37) MLYCDC5AR1F10
SCHEMBL3581186 0.89 CNR1 (0.39) C5AR1TRPV1CYP2C19
SCHEMBL3579944 0.88 MCHR1 (0.39) MLYCDTRPM8OPRM1OPRD1C5AR1
SCHEMBL3573512 0.86 HDAC1 (0.36) SIGMAR1HSP90AA1OPRM1OPRD1C5AR1
SCHEMBL3581889 0.85 C5AR1 (0.40) C5AR1F10KLKB1
SCHEMBL3580029 0.85 MLYCD (0.34) MLYCDSIGMAR1HSP90AA1OPRM1OPRD1
SCHEMBL1397638 0.84 HCRTR1 (0.37) SIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7678818-B2 Anthranilamide and 2-amino-heteroarene-carboxamide compounds HOFFMANN-LA ROCHE INC. (US) 2010-03-16 US claimed
EP-1984340-B1 ANTHRANILAMIDE/2-AMINO-HETEROARENE CARBOXAMIDE DERIVATIVES HOFFMANN LA ROCHE (CH) 2012-06-27 EP disclosed