SCHEMBL3584062

SCHEMBL3584062

CNc1ncc(Br)cc1C(=O)N(CCc1ccc(Cl)c(Cl)c1)Cc1ccc(C(F)(C(F)(F)F)C(F)(F)F)cc1

nearest known ligand 0.35

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
GBA1 P04062 3/20 0.34
HSP90AA1 P07900 2/20 0.34
SSTR2 P30874 6/20 0.34
SSTR4 P31391 6/20 0.34
MLYCD O95822 1/20 0.33
CENPE Q02224 2/20 0.33
SIGMAR1 Q99720 1/20 0.32
OPRM1 P35372 1/20 0.32
OPRD1 P41143 1/20 0.32
CETP P11597 1/20 0.32
RAF1 P04049 1/20 0.32
MAP2K1 Q02750 1/20 0.32
TRPV1 Q8NER1 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3574238 0.92 MLYCD (0.35) HSP90AA1MLYCDCENPESIGMAR1OPRM1
SCHEMBL3584126 0.91 ESRRG (0.36) GBA1HSP90AA1SSTR2SSTR4SIGMAR1
SCHEMBL3569329 0.84 C5AR1 (0.41) MLYCD
SCHEMBL3576692 0.83 ESRRG (0.37) HSP90AA1SIGMAR1OPRM1OPRD1TRPV1
SCHEMBL3580029 0.83 MLYCD (0.34) HSP90AA1MLYCDCENPESIGMAR1OPRM1
SCHEMBL3579477 0.82 MCHR1 (0.37) MLYCD
SCHEMBL3578672 0.82 GBA1 (0.34) GBA1HSP90AA1SSTR2SSTR4SIGMAR1
SCHEMBL3575573 0.82 HSP90AA1 (0.36) GBA1HSP90AA1SSTR2SSTR4OPRM1
SCHEMBL3574285 0.82 ESRRG (0.36) HSP90AA1CENPESIGMAR1OPRM1OPRD1
SCHEMBL3581186 0.81 CNR1 (0.39) TRPV1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7678818-B2 Anthranilamide and 2-amino-heteroarene-carboxamide compounds HOFFMANN-LA ROCHE INC. (US) 2010-03-16 US claimed
EP-2654751-A1 PHOSPHORUS-SUBSTITUTED QUINOXALINE-TYPE PIPERIDINE COMPOUNDS AND USES THEREOF Purdue Pharma L.P. (US) 2013-10-30 EP disclosed
WO-2012085648-A9 PHOSPHORUS-SUBSTITUTED QUINOXALINE-TYPE PIPERIDINE COMPOUNDS AND USES THEREOF PURDUE PHARMA L.P. (US) 2013-03-21 WO disclosed
WO-2012085648-A1 PHOSPHORUS-SUBSTITUTED QUINOXALINE-TYPE PIPERIDINE COMPOUNDS AND USES THEREOF PURDUE PHARMA L.P. (US) 2012-06-28 WO disclosed
EP-1984340-B1 ANTHRANILAMIDE/2-AMINO-HETEROARENE CARBOXAMIDE DERIVATIVES HOFFMANN LA ROCHE (CH) 2012-06-27 EP disclosed