SCHEMBL3580029

SCHEMBL3580029

CNc1cnc(Cl)cc1C(=O)N(CCc1ccc(Cl)c(Cl)c1)Cc1ccc(C(F)(C(F)(F)F)C(F)(F)F)cc1

nearest known ligand 0.36

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
MLYCD O95822 1/20 0.34
SIGMAR1 Q99720 2/20 0.33
HSP90AA1 P07900 2/20 0.33
OPRM1 P35372 1/20 0.33
OPRD1 P41143 1/20 0.33
RAF1 P04049 1/20 0.33
MAP2K1 Q02750 1/20 0.33
TRPV1 Q8NER1 1/20 0.32
KCNH2 Q12809 2/20 0.32
TMEM97 Q5BJF2 2/20 0.32
CENPE Q02224 2/20 0.31
CYP2C19 P33261 1/20 0.31
RPS6KB1 P23443 1/20 0.31
LIPC P11150 1/20 0.31
LIPG Q9Y5X9 1/20 0.31
C5AR1 P21730 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3574969 0.91 C5AR1 (0.39) MLYCDHSP90AA1C5AR1
SCHEMBL3574044 0.90 NR1H4 (0.37) SIGMAR1HSP90AA1OPRM1OPRD1
SCHEMBL3575504 0.89 SLC2A1 (0.38) TRPV1CYP2C19
SCHEMBL3574238 0.85 MLYCD (0.35) MLYCDSIGMAR1HSP90AA1OPRM1OPRD1
SCHEMBL3577889 0.84 C5AR1 (0.39) MLYCDHSP90AA1C5AR1
SCHEMBL1397709 0.83 OPRM1 (0.35) SIGMAR1OPRM1OPRD1RAF1MAP2K1
SCHEMBL3584062 0.83 GBA1 (0.34) MLYCDSIGMAR1HSP90AA1OPRM1OPRD1
SCHEMBL3581176 0.82 SLC2A1 (0.38) TRPV1CYP2C19
SCHEMBL3584245 0.82 SIGMAR1 (0.34) SIGMAR1OPRM1OPRD1CYP2C19LIPG
SCHEMBL3579370 0.81 SLC2A1 (0.39) TRPV1CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7678818-B2 Anthranilamide and 2-amino-heteroarene-carboxamide compounds HOFFMANN-LA ROCHE INC. (US) 2010-03-16 US claimed
EP-1984340-B1 ANTHRANILAMIDE/2-AMINO-HETEROARENE CARBOXAMIDE DERIVATIVES HOFFMANN LA ROCHE (CH) 2012-06-27 EP disclosed