SCHEMBL3574285

SCHEMBL3574285

CNc1ncc(F)cc1C(=O)N(CCc1ccc(Cl)c(Cl)c1)Cc1ccc(C(C)(C)C)cc1

nearest known ligand 0.36

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ESRRG P62508 2/20 0.36
NR1H4 Q96RI1 1/20 0.36
TP53 P04637 1/20 0.36
MAPT P10636 1/20 0.36
CENPE Q02224 8/20 0.35
ESRRB O95718 1/20 0.35
NR1I3 Q14994 1/20 0.35
TRPM8 Q7Z2W7 1/20 0.34
SIGMAR1 Q99720 1/20 0.34
HSP90AA1 P07900 1/20 0.34
OPRM1 P35372 1/20 0.33
OPRD1 P41143 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3583608 0.91 ESRRG (0.35) ESRRGNR1H4TP53MAPTCENPE
SCHEMBL3576692 0.91 ESRRG (0.37) ESRRGNR1H4ESRRBNR1I3TRPM8
SCHEMBL3580374 0.90 ESRRG (0.36) ESRRGNR1H4TP53MAPTESRRB
SCHEMBL3584126 0.89 ESRRG (0.36) ESRRGNR1H4ESRRBNR1I3SIGMAR1
SCHEMBL3587153 0.89 ESRRG (0.36) ESRRGNR1H4TP53MAPTESRRB
SCHEMBL3576972 0.89 BTK (0.36) ESRRGNR1H4TP53MAPTCENPE
SCHEMBL9958256 0.89 NR1H4 (0.38) ESRRGNR1H4TP53MAPTCENPE
SCHEMBL3580346 0.88 ESRRG (0.35) ESRRGNR1H4ESRRBNR1I3TRPM8
SCHEMBL3586398 0.87 PTGES (0.39) ESRRGNR1H4NR1I3OPRM1OPRD1
SCHEMBL3580658 0.85 RAF1 (0.39) ESRRGNR1H4ESRRBSIGMAR1HSP90AA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7678818-B2 Anthranilamide and 2-amino-heteroarene-carboxamide compounds HOFFMANN-LA ROCHE INC. (US) 2010-03-16 US claimed
EP-1984340-B1 ANTHRANILAMIDE/2-AMINO-HETEROARENE CARBOXAMIDE DERIVATIVES HOFFMANN LA ROCHE (CH) 2012-06-27 EP disclosed