SCHEMBL3584126

SCHEMBL3584126

CNc1ncc(Br)cc1C(=O)N(CCc1ccc(Cl)c(Cl)c1)Cc1ccc(C(C)(C)C)cc1

nearest known ligand 0.36

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ESRRG P62508 2/20 0.36
GBA1 P04062 3/20 0.36
NR1H4 Q96RI1 1/20 0.36
HSP90AA1 P07900 2/20 0.35
ESRRB O95718 1/20 0.35
SSTR2 P30874 5/20 0.35
SSTR4 P31391 5/20 0.35
NR1I3 Q14994 1/20 0.35
SIGMAR1 Q99720 1/20 0.34
OPRM1 P35372 1/20 0.33
OPRD1 P41143 1/20 0.33
HDAC3 O15379 1/20 0.33
HDAC8 Q9BY41 1/20 0.33
HDAC6 Q9UBN7 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3575573 0.91 HSP90AA1 (0.36) ESRRGGBA1NR1H4HSP90AA1ESRRB
SCHEMBL3576692 0.91 ESRRG (0.37) ESRRGNR1H4HSP90AA1ESRRBNR1I3
SCHEMBL3584062 0.91 GBA1 (0.34) GBA1HSP90AA1SSTR2SSTR4SIGMAR1
SCHEMBL3580374 0.90 ESRRG (0.36) ESRRGNR1H4HSP90AA1ESRRBNR1I3
SCHEMBL3587153 0.89 ESRRG (0.36) ESRRGNR1H4HSP90AA1ESRRBNR1I3
SCHEMBL3574285 0.89 ESRRG (0.36) ESRRGNR1H4HSP90AA1ESRRBNR1I3
SCHEMBL9957773 0.89 NR1H4 (0.38) ESRRGGBA1NR1H4HSP90AA1ESRRB
SCHEMBL3580346 0.88 ESRRG (0.35) ESRRGNR1H4HSP90AA1ESRRBNR1I3
SCHEMBL3586398 0.87 PTGES (0.39) ESRRGNR1H4NR1I3OPRM1OPRD1
SCHEMBL3580658 0.85 RAF1 (0.39) ESRRGNR1H4HSP90AA1ESRRBSIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7678818-B2 Anthranilamide and 2-amino-heteroarene-carboxamide compounds HOFFMANN-LA ROCHE INC. (US) 2010-03-16 US claimed
EP-1984340-B1 ANTHRANILAMIDE/2-AMINO-HETEROARENE CARBOXAMIDE DERIVATIVES HOFFMANN LA ROCHE (CH) 2012-06-27 EP disclosed