SCHEMBL3580346

SCHEMBL3580346

C=Cc1cnc(NC)c(C(=O)N(CCc2ccc(Cl)c(Cl)c2)Cc2ccc(C(C)(C)C)cc2)c1

nearest known ligand 0.35

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ESRRG P62508 2/20 0.35
NR1H4 Q96RI1 1/20 0.35
ESRRB O95718 1/20 0.34
NR1I3 Q14994 1/20 0.34
HSP90AA1 P07900 2/20 0.33
VNN1 O95497 1/20 0.33
SIGMAR1 Q99720 1/20 0.33
OPRM1 P35372 1/20 0.33
OPRD1 P41143 1/20 0.33
TRPM8 Q7Z2W7 1/20 0.32
KCNH2 Q12809 2/20 0.31
CYP2C19 P33261 2/20 0.31
TRPV1 Q8NER1 1/20 0.31
CYP1A2 P05177 1/20 0.31
CYP3A4 P08684 1/20 0.31
CYP2D6 P10635 1/20 0.31
CYP2C9 P11712 1/20 0.31
MAPK1 P28482 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3576692 0.89 ESRRG (0.37) ESRRGNR1H4ESRRBNR1I3HSP90AA1
SCHEMBL3580374 0.89 ESRRG (0.36) ESRRGNR1H4ESRRBNR1I3HSP90AA1
SCHEMBL3587153 0.88 ESRRG (0.36) ESRRGNR1H4ESRRBNR1I3HSP90AA1
SCHEMBL3584126 0.88 ESRRG (0.36) ESRRGNR1H4ESRRBNR1I3HSP90AA1
SCHEMBL3574285 0.88 ESRRG (0.36) ESRRGNR1H4ESRRBNR1I3HSP90AA1
SCHEMBL3586398 0.85 PTGES (0.39) ESRRGNR1H4NR1I3OPRM1OPRD1
SCHEMBL3580658 0.84 RAF1 (0.39) ESRRGNR1H4ESRRBHSP90AA1SIGMAR1
SCHEMBL1397638 0.81 HCRTR1 (0.37) NR1I3SIGMAR1
SCHEMBL3574238 0.81 MLYCD (0.35) HSP90AA1SIGMAR1OPRM1OPRD1TRPM8
SCHEMBL3585932 0.81 CCR9 (0.36) ESRRGNR1H4ESRRBNR1I3HSP90AA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7678818-B2 Anthranilamide and 2-amino-heteroarene-carboxamide compounds HOFFMANN-LA ROCHE INC. (US) 2010-03-16 US claimed
EP-1984340-B1 ANTHRANILAMIDE/2-AMINO-HETEROARENE CARBOXAMIDE DERIVATIVES HOFFMANN LA ROCHE (CH) 2012-06-27 EP disclosed