SCHEMBL3580405

SCHEMBL3580405

CCOC(=O)c1cccc2nc(-c3ccc([N+](=O)[O-])cc3)[nH]c12

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MMP2 P08253 3/20 0.50
MMP9 P14780 3/20 0.50
MMP8 P22894 3/20 0.50
AR P10275 2/20 0.50
PARP1 P09874 3/20 0.48
RAB9A P51151 3/20 0.48
GAA P10253 1/20 0.48
MAPT P10636 5/20 0.47
TNKS O95271 2/20 0.47
TNKS2 Q9H2K2 2/20 0.47
GUSB P08236 1/20 0.47
NLRP3 Q96P20 1/20 0.47
PARP2 Q9UGN5 1/20 0.47
NPBWR1 P48145 2/20 0.47
MMP13 P45452 2/20 0.46
MEN1 O00255 2/20 0.46
KMT2A Q03164 2/20 0.46
POLB P06746 1/20 0.46
ALDH1A1 P00352 2/20 0.46
DGAT1 O75907 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3574926 0.89 MAPT (0.55) MMP2MMP9MMP8RAB9AMAPT
SCHEMBL6948237 0.85 TSHR (0.50) PARP1RAB9AGAAMAPTMEN1
SCHEMBL6810427 0.83 PKN1 (0.58) MMP2PARP1MMP13MAPK1
SCHEMBL3580402 0.83 PARP1 (0.69) MMP2MMP9MMP8ARPARP1
SCHEMBL6330688 0.79 MMP2 (0.62) MMP2MMP9MMP8PARP1RAB9A
SCHEMBL6170666 0.78 TSHR (0.53) PARP1GAAMAPTPOLBALDH1A1
SCHEMBL6804379 0.78 ATM (0.52) PARP1MAPTMEN1KMT2APOLB
SCHEMBL3575168 0.77 SIRT2 (0.52) PARP1GAAMAPTTNKSTNKS2
SCHEMBL3580810 0.76 CHEK1 (0.59) PARP1RAB9AGAAGUSBPOLB
SCHEMBL3577856 0.76 KDM4E (0.50) PARP1RAB9AMAPTMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7781596-B1 Substituted 2-phenylbenzimidazoles, the production thereof and their use ABBOTT LABORATORIES (US) 2010-08-24 US disclosed