SCHEMBL3584976

SCHEMBL3584976

Cc1cc(N2CCNCC2)ccc1-c1nc2cccc(C(N)=O)c2[nH]1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ACVR1 Q04771 6/20 0.42
JAK2 O60674 1/20 0.42
ADRB1 P08588 2/20 0.41
TGFBR1 P36897 2/20 0.41
HTR1A P08908 1/20 0.41
HTR7 P34969 1/20 0.41
PIM1 P11309 1/20 0.40
PIM3 Q86V86 1/20 0.40
PIM2 Q9P1W9 1/20 0.40
PDE7A Q13946 2/20 0.40
TGFB2 P61812 1/20 0.40
PDE4D Q08499 1/20 0.39
PDE7B Q9NP56 1/20 0.39
PARP1 P09874 1/20 0.39
AURKA O14965 1/20 0.38
AURKB Q96GD4 1/20 0.38
CYP1A2 P05177 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2D6 P10635 1/20 0.38
TSHR P16473 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3584970 0.84 PARP1 (0.53) PIM1PARP1AURKAAURKBCLK4
SCHEMBL3582864 0.83 GRK6 (0.48) JAK2ADRB1HTR1AHTR7PARP1
SCHEMBL3580358 0.83 PARP1 (0.53) ACVR1JAK2TGFBR1PIM1PIM3
SCHEMBL3582373 0.82 PARP1 (0.49) ACVR1PIM1PIM3PIM2PARP1
SCHEMBL5621810 0.76 HTR3A (0.52) PARP1AURKACLK4
SCHEMBL5621910 0.74 HTR3A (0.48) PIM1PARP1
SCHEMBL1741562 0.74 ADRB1 (0.61) ACVR1ADRB1TGFBR1HTR1AHTR7
SCHEMBL30798753 0.74 ADRB1 (0.61) ACVR1ADRB1TGFBR1HTR1AHTR7
SCHEMBL6582942 0.74 PARP1 (0.43) ACVR1ADRB1TGFBR1HTR7PIM1
SCHEMBL3587289 0.74 AURKA (0.56) JAK2PARP1AURKAAURKBCHEK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7781596-B1 Substituted 2-phenylbenzimidazoles, the production thereof and their use ABBOTT LABORATORIES (US) 2010-08-24 US disclosed