SCHEMBL3586495

SCHEMBL3586495

COc1ccc(-c2nc3cccc(C(N)=O)c3[nH]2)cc1OCCN(C)C

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 3/20 0.56
ADORA1 P30542 2/20 0.56
MAP4K4 O95819 2/20 0.53
PIM1 P11309 2/20 0.53
PIM3 Q86V86 2/20 0.53
AURKB Q96GD4 2/20 0.53
CLK4 Q9HAZ1 2/20 0.53
STK17A Q9UEE5 2/20 0.53
MAP4K5 Q9Y4K4 2/20 0.53
DYRK3 O43781 1/20 0.53
RPS6KB1 P23443 1/20 0.53
CSNK2A1 P68400 1/20 0.53
PKN2 Q16513 1/20 0.53
BRSK1 Q8TDC3 1/20 0.53
HIPK2 Q9H2X6 1/20 0.53
MKNK2 Q9HBH9 1/20 0.53
PARP1 P09874 7/20 0.53
PDE4A P27815 2/20 0.47
PDE4B Q07343 2/20 0.47
PDE4C Q08493 2/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3577822 0.85 MAP4K4 (0.72) ADORA2AADORA1MAP4K4PIM1PIM3
SCHEMBL3586486 0.85 PARP1 (0.76) MAP4K4PIM1PIM3AURKBCLK4
SCHEMBL3582880 0.82 ALDH1A1 (0.47) ADORA1MAP4K4PIM1PIM3AURKB
SCHEMBL6805384 0.79 CLK4 (0.44) MAP4K4PIM1PIM3AURKBCLK4
SCHEMBL4740751 0.78 GUSB (0.59) PARP1PDE4APDE4BPDE4CPDE4D
SCHEMBL7137103 0.78 PARP1 (0.55) MAP4K4PIM1PIM3AURKBCLK4
SCHEMBL7131933 0.77 PARP1 (0.54) MAP4K4PIM1PIM3AURKBCLK4
SCHEMBL6584505 0.76 MAP4K4 (0.57) ADORA2AADORA1MAP4K4PIM1PIM3
SCHEMBL31053400 0.76 PARP1 (0.67) MAP4K4PIM1PIM3AURKBCLK4
SCHEMBL3577456 0.76 MAP4K4 (0.59) ADORA2AADORA1MAP4K4PIM1PIM3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7781596-B1 Substituted 2-phenylbenzimidazoles, the production thereof and their use ABBOTT LABORATORIES (US) 2010-08-24 US disclosed