SCHEMBL359222

SCHEMBL359222

COCCOc1cnc2ccc(CC=O)cc2c1

nearest known ligand 0.47

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
MET P08581 9/20 0.47
CBFB Q13951 2/20 0.41
ALDH1A1 P00352 1/20 0.41
F2 P00734 1/20 0.41
GLA P06280 1/20 0.41
HPGD P15428 1/20 0.41
CYP3A4 P08684 1/20 0.39
PDGFRB P09619 3/20 0.39
PDGFRA P16234 3/20 0.39
APP P05067 1/20 0.37
PDE10A Q9Y233 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL187290 0.83 CBFB (0.57) METCBFBALDH1A1F2GLA
SCHEMBL186997 0.82 FDPS (0.43) METCBFBALDH1A1F2GLA
SCHEMBL370132 0.81 CBFB (0.46) METCBFBALDH1A1F2GLA
SCHEMBL187431 0.77 FBP1 (0.44) METCBFBALDH1A1F2GLA
SCHEMBL358693 0.77 CNR1 (0.47) METCBFBALDH1A1F2GLA
SCHEMBL358992 0.77 EGFR (0.42) METCBFBALDH1A1F2GLA
SCHEMBL13619702 0.77 MET (0.42) METCBFBALDH1A1F2GLA
SCHEMBL359885 0.77 MET (0.42) METCBFBALDH1A1F2GLA
SCHEMBL2698219 0.77 ALDH1A1 (0.43) METCBFBALDH1A1F2GLA
SCHEMBL186985 0.77 PDGFRB (0.43) METCBFBALDH1A1F2GLA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2593107-A1 TYROSINE KINASE INHIBITORS Merck Sharp & Dohme Corp. (US) 2013-05-22 EP disclosed
WO-2012009194-A1 TYROSINE KINASE INHIBITORS MERCK SHARP & DOHME CORP. (US) 2012-01-19 WO disclosed