SCHEMBL3593028

SCHEMBL3593028

CC(N)c1c(-c2ccc(Cl)cc2Cl)ncn1Cc1ccccc1

nearest known ligand 0.50

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.44
GAA P10253 1/20 0.44
HPGD P15428 1/20 0.44
CXCR2 P25025 1/20 0.41
CNR1 P21554 3/20 0.41
MDM4 O15151 2/20 0.40
TP53 P04637 2/20 0.40
MDM2 Q00987 2/20 0.40
DPP4 P27487 7/20 0.40
DPP8 Q6V1X1 3/20 0.40
CYP3A4 P08684 4/20 0.39
CYP2C19 P33261 3/20 0.39
DPP9 Q86TI2 2/20 0.39
KCNH2 Q12809 1/20 0.39
MARS1 P56192 1/20 0.38
HSD11B1 P28845 1/20 0.38
CRHR1 P34998 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3594733 0.90 CXCR2 (0.44) ALDH1A1GAAHPGDCXCR2CNR1
SCHEMBL3600972 0.89 DPP4 (0.41) ALDH1A1GAAHPGDCNR1MDM4
SCHEMBL3592478 0.89 P2RX7 (0.44) ALDH1A1MDM4MDM2DPP4DPP8
SCHEMBL3605612 0.88 CNR1 (0.43) CNR1DPP4DPP8CYP3A4CYP2C19
SCHEMBL3597273 0.88 CXCR2 (0.40) ALDH1A1GAAHPGDCXCR2CNR1
SCHEMBL3595008 0.87 CXCR2 (0.50) CXCR2TP53DPP4
SCHEMBL3599359 0.87 CXCR2 (0.40) ALDH1A1GAAHPGDCXCR2CNR1
SCHEMBL3598037 0.86 CXCR2 (0.47) ALDH1A1CXCR2CNR1TP53DPP4
SCHEMBL3600416 0.86 CNR1 (0.42) CNR1MDM4MDM2DPP4DPP8
SCHEMBL3602324 0.86 CYP11B1 (0.41) ALDH1A1GAAHPGDCNR1TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7728146-B2 Enzyme inhibitors PROBIODRUG AG (DE) 2010-06-01 US claimed