SCHEMBL360387

SCHEMBL360387

COc1ccc(NC(N)=O)cc1

nearest known ligand 0.70

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 5/20 0.70
RAB9A P51151 5/20 0.70
SMN1; SMN2 Q16637 4/20 0.70
ALDH1A1 P00352 1/20 0.65
GLA P06280 1/20 0.65
TP53 P04637 2/20 0.63
ALOX15 P16050 1/20 0.63
TGM2 P21980 1/20 0.59
L3MBTL1 Q9Y468 1/20 0.59
MAPT P10636 3/20 0.58
KDM4E B2RXH2 1/20 0.58
MEN1 O00255 1/20 0.58
KMT2A Q03164 1/20 0.58
SAE1 Q9UBE0 1/20 0.58
UBA2 Q9UBT2 1/20 0.58
CYP1A2 P05177 1/20 0.58
CYP2D6 P10635 1/20 0.58
CYP2C9 P11712 1/20 0.58
HPGD P15428 1/20 0.58
CYP2C19 P33261 1/20 0.58

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12845568 0.94 KIF11 (0.65) NPC1RAB9ASMN1; SMN2ALDH1A1GLA
SCHEMBL6152116 0.85 KMT2A (0.74) NPC1RAB9ASMN1; SMN2ALDH1A1L3MBTL1
SCHEMBL4087493 0.84 RAB9A (0.66) NPC1RAB9ASMN1; SMN2ALDH1A1TP53
SCHEMBL29673494 0.84 ALDH1A1 (0.59) NPC1RAB9ASMN1; SMN2ALDH1A1MAPT
SCHEMBL11092496 0.83 RAB9A (1.00) NPC1RAB9ASMN1; SMN2TP53ALOX15
SCHEMBL6396790 0.83 RAB9A (0.76) NPC1RAB9ASMN1; SMN2ALDH1A1TP53
SCHEMBL31090324 0.82 GAA (0.62) NPC1RAB9ASMN1; SMN2ALDH1A1MAPT
SCHEMBL4105580 0.82 NPC1 (0.58) NPC1RAB9ASMN1; SMN2ALDH1A1GLA
SCHEMBL29484162 0.82 MAPK1 (0.62) NPC1RAB9ASMN1; SMN2ALDH1A1TP53
SCHEMBL5062623 0.82 PEPD (0.80) NPC1RAB9AALDH1A1GLAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 386 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113906321-B Polarizing plate, method for manufacturing same, and image display device 住友化学株式会社 2024-10-15 CN claimed
US-20240262801-A1 COMPOUNDS HAVING 5-(2-FLUORO-6-HYDROXYPHENYL)-1,2,5-THIADIAZOLIDIN-3-ONE 1,1-DIOXIDE AS INHIBITORS OF PROTEIN KINASE PHOSPHATASE ENZYMES MONDEGO BIO, LDA. (PT) 2024-08-08 US claimed
US-12018021-B2 Thiophene derivatives for the treatment of disorders caused by IgE UCB Biopharma SRL (BE) 2024-06-25 US claimed
CN-115926228-B Protective layer, preparation method thereof and lithium ion battery 蜂巢能源科技(无锡)有限公司 2024-05-31 CN claimed
CN-117946033-A Preparation method for photo-promoted synthesis of urea compound 兰州大学 2024-04-30 CN claimed
CN-115926228-A Protective layer, preparation method thereof and lithium ion battery 蜂巢能源科技(无锡)有限公司 2023-04-07 CN claimed
CN-111303554-B PVC plastic and preparation method thereof 温州市隆昌塑料有限公司 2022-06-14 CN claimed
CN-114057499-A Sliding plate brick and preparation method thereof 江苏盛耐新材料有限公司 2022-02-18 CN claimed
EP-3810606-A1 THIOPHENE DERIVATIVES FOR THE TREATMENT OF DISORDERS CAUSED BY IGE UCB Biopharma SRL (BE) 2021-04-28 EP claimed
CN-112566910-A Thiophene derivatives for the treatment of IgE induced diseases UCB生物制药有限责任公司 2021-03-26 CN claimed
EP-1118322-A1 DRUGS FOR IMPROVING VESICAL EXCRETORY STRENGTH Takeda Chemical Industries, Ltd. (JP) 2001-07-25 EP claimed
EP-0858455-A4 4-OXA AND 4-THIA STEROIDS MERCK & CO INC (US) 2000-04-12 EP claimed
US-5998464-A 4-Oxa and 4-thia steroids MERCK & CO., INC. (US) 1999-12-07 US claimed
US-5817802-A IN IONIZING MEDIUM WITH A TRIALKYLSILANE MERCK & CO., INC. (US) 1998-10-06 US claimed
EP-0858455-A1 4-OXA AND 4-THIA STEROIDS Merck & Co., Inc. (US) 1998-08-19 EP claimed
US-5777134-A 4-oxa and 4-thia steriods MERCK & CO., INC. (US) 1998-07-07 US claimed
US-5696266-A HYDROGENATING DELTA-5-STEROIDAL ENELACTAM DISSOLVED IN SOLVENT IN PRESENCE OF RHODIUM CATALYST MERCK & CO., INC. (US) 1997-12-09 US claimed
WO-1997015564-A1 4-OXA AND 4-THIA STEROIDS MERCK & CO., INC. (US) 1997-05-01 WO claimed
WO-1996007643-A1 PROCESS FOR THE STEREOSELECTIVE REDUCTION OF STEROID ENELACTAMS MERCK & CO., INC. (US) 1996-03-14 WO claimed
US-4285863-A YELLOW-TO-RED ORGANIC PIGMENTS; PLASTICS AND FABRICS; PAINTS, ENAMELS, AND INKS MONTEDISON S.P.A. (IT) 1981-08-25 US claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20240262801-A1 COMPOUNDS HAVING 5-(2-FLUORO-6-HYDROXYPHENYL)-1,2,5-THIADIAZOLIDIN-3-ONE 1,1-DIOXIDE AS INHIBITORS OF PROTEIN KINASE PHOSPHATASE ENZYMES PPM1A, TH, PPM1G NPC1 2925/4885RAB9A 2110/4885SMN1; SMN2 3686/4885
US-12018021-B2 Thiophene derivatives for the treatment of disorders caused by IgE TSLP, CYSLTR1, CYSLTR2 NPC1 185/4885RAB9A 2032/4885SMN1; SMN2 4377/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.