SCHEMBL3605764

SCHEMBL3605764

CC(C)(C)[Si](C)(C)OCc1cccc(OC[C@@H]2CCCCN2C(=O)O)n1

nearest known ligand 0.39

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 4/20 0.39
NPC1 O15118 2/20 0.39
ABHD6 Q9BV23 3/20 0.38
DAGLA Q9Y4D2 3/20 0.38
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
CNR2 P34972 1/20 0.37
LMNA P02545 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
HCRTR2 O43614 5/20 0.36
CYP2D6 P10635 1/20 0.35
DPP4 P27487 1/20 0.35
DPP8 Q6V1X1 1/20 0.35
DPP9 Q86TI2 1/20 0.35
DPP7 Q9UHL4 1/20 0.35
HPGD P15428 1/20 0.35
SPHK2 Q9NRA0 1/20 0.35
ALDH1A1 P00352 1/20 0.35
NR2F2 P24468 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3607859 0.97 CYP2D6 (0.38) RAB9ANPC1ABHD6DAGLAMEN1
SCHEMBL3615900 0.83 CNR2 (0.42) RAB9ANPC1ABHD6DAGLAMEN1
SCHEMBL3608576 0.83 DAGLB (0.43) RAB9ANPC1ABHD6DAGLAMEN1
SCHEMBL3602873 0.80 DAGLB (0.40) ABHD6DAGLACNR2CYP2D6DPP4
SCHEMBL3606003 0.80 CNR2 (0.40) ABHD6DAGLACNR2CYP2D6DPP4
SCHEMBL3602535 0.74 HRH3 (0.37) KMT2A
SCHEMBL4566643 0.74 KCNH2 (0.33)
SCHEMBL3637452 0.71 FKBP1A (0.48) ABHD6DAGLA
SCHEMBL30369514 0.71 HCRTR1 (0.37) RAB9ANPC1HCRTR2HPGDALDH1A1
SCHEMBL17008464 0.70 ABHD6 (0.58) RAB9ANPC1ABHD6DAGLAHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7723331-B2 Thienopyrimidine compounds and uses thereof ASTRAZENECA AB (SE) 2010-05-25 US disclosed
US-20080051405-A1 Therapeutic Agents ASTRAZENECA AB (SE) 2008-02-28 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080051405-A1 Therapeutic Agents GPR119, HTT, IAPP RAB9A 1071/4885NPC1 148/4885ABHD6 1481/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.