SCHEMBL3607558

SCHEMBL3607558

COCCOC(=O)Nc1c(C)cc(Br)cc1C

nearest known ligand 0.49

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
MAPT P10636 1/20 0.49
NLRP3 Q96P20 2/20 0.47
ALDH1A1 P00352 4/20 0.46
HPGD P15428 1/20 0.43
LCK P06239 1/20 0.41
TAS1R3 Q7RTX0 1/20 0.40
TAS1R1 Q7RTX1 1/20 0.40
TAS1R2 Q8TE23 1/20 0.40
MAPK1 P28482 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.38
KDM4E B2RXH2 3/20 0.38
PKM P14618 1/20 0.38
KMT2A Q03164 2/20 0.38
CSNK2A2 P19784 1/20 0.38
CSNK2A1 P68400 1/20 0.38
MEN1 O00255 1/20 0.38
GPR35 Q9HC97 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3106554 0.86 MAPK1 (0.52) MAPTNLRP3ALDH1A1HPGDTAS1R3
SCHEMBL1000325 0.83 NLRP3 (0.59) MAPTNLRP3ALDH1A1HPGDTAS1R3
SCHEMBL3600751 0.82 NLRP3 (0.48) NLRP3HPGDMAPK1SMN1; SMN2KDM4E
SCHEMBL31059176 0.81 MAPT (0.54) MAPTNLRP3ALDH1A1HPGDLCK
SCHEMBL25307579 0.73 NLRP3 (0.48) MAPTNLRP3ALDH1A1HPGDMAPK1
SCHEMBL30201354 0.73 NLRP3 (0.48) MAPTNLRP3ALDH1A1HPGDMAPK1
SCHEMBL29413069 0.73 NLRP3 (0.48) MAPTNLRP3ALDH1A1HPGDSMN1; SMN2
SCHEMBL25243093 0.72 LCK (0.62) MAPTALDH1A1HPGDLCKTAS1R3
SCHEMBL30487417 0.72 ALDH1A1 (0.54) MAPTALDH1A1HPGDLCKTAS1R3
SCHEMBL18415477 0.72 ALDH1A1 (0.61) MAPTALDH1A1HPGDLCKTAS1R3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8835476-B2 Synthesis of novel antimicrobials WU FAN (CA) 2014-09-16 US disclosed
US-20100076028-A1 Design and Synthesis of Novel Antimicrobials WU FAN 2010-03-25 US disclosed
US-20100063044-A1 SUBSTITUTED ANILINE DERIVATIVES H. LUNDBECK A/S (DK) 2010-03-11 US disclosed
US-7601870-B2 Such as Hexanoic acid (4-bromo-2,6-dimethyl-phenyl)-amide; potassium channel modulators; epilepsy H. LUNDBECK A/S (DK) 2009-10-13 US disclosed
EP-1791809-A1 SUBSTITUTED ANILINE DERIVATIVES H. LUNDBECK A/S (DK) 2007-06-06 EP disclosed
US-20060155121-A1 Substituted aniline derivatives H. LUNDBECK A/S (DK) 2006-07-13 US disclosed
WO-2006029623-A1 SUBSTITUTED ANILINE DERIVATIVES H. LUNDBECK A/S (DK) 2006-03-23 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100063044-A1 SUBSTITUTED ANILINE DERIVATIVES NDUFS3, NAT1, PRMT3 MAPT 2817/4885NLRP3 3233/4885ALDH1A1 206/4885
US-20100076028-A1 Design and Synthesis of Novel Antimicrobials MLX, LPXN, TPX2 MAPT 4883/4885NLRP3 642/4885ALDH1A1 4295/4885
US-20060155121-A1 Substituted aniline derivatives UGT2B7, NAT1, CYP1A2 MAPT 1406/4885NLRP3 4464/4885ALDH1A1 178/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.