SCHEMBL3625399

SCHEMBL3625399

COc1ccc2c(O)cc(-c3nc(C(C)C)oc3C)nc2c1C

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.35
HPGD P15428 4/20 0.35
HSD17B10 Q99714 4/20 0.35
KDM4E B2RXH2 4/20 0.35
TSHR P16473 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
ESR1 P03372 2/20 0.34
ESR2 Q92731 2/20 0.34
MCL1 Q07820 5/20 0.34
HIF1A Q16665 2/20 0.33
MAPT P10636 3/20 0.33
NPC1 O15118 2/20 0.33
RAB9A P51151 1/20 0.33
CA12 O43570 3/20 0.31
CA1 P00915 3/20 0.31
CA7 P43166 3/20 0.31
CA9 Q16790 3/20 0.31
CA13 Q8N1Q1 3/20 0.31
AKR1B1 P15121 2/20 0.31
LMNA P02545 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2624139 0.76 GPR35 (0.36) ALDH1A1HPGDHSD17B10KDM4ETSHR
SCHEMBL997481 0.75 ADORA2A (0.33) ALDH1A1NPC1NPSR1POLBMEN1
SCHEMBL3627208 0.74 TDO2 (0.51) ALDH1A1HPGDHSD17B10KDM4ETSHR
SCHEMBL13226974 0.74 RAC1 (0.32) KDM4EMAPTNPC1RAB9ANPSR1
SCHEMBL313693 0.74 CTSS (0.38) ALDH1A1HSD17B10KDM4ETSHRL3MBTL1
SCHEMBL3625396 0.73 HTT (0.36) ALDH1A1HPGDHSD17B10KDM4ETSHR
SCHEMBL3624833 0.73 ENPP3 (0.43) ALDH1A1HPGDHSD17B10KDM4ETSHR
SCHEMBL16064009 0.73 TDO2 (0.33) ALDH1A1HPGDHSD17B10KDM4EL3MBTL1
SCHEMBL996497 0.72 CCR1 (0.42) MAPTNPC1RAB9ALMNAMEN1
SCHEMBL3659800 0.71 MEN1 (0.34) ALDH1A1HPGDHSD17B10KDM4ETSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010033466-A1 MACROCYCLIC INHIBITORS OF HEPATITIS C PROTEASE PHENOMIX CORPORATION (US) 2010-03-25 WO disclosed