SCHEMBL362986

SCHEMBL362986

Cc1nc2ccccc2c2ccnn12

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR3E A5X5Y0 1/20 0.56
HTR3B O95264 1/20 0.56
HTR3A P46098 1/20 0.56
HTR3D Q70Z44 1/20 0.56
HTR3C Q8WXA8 1/20 0.56
KDM4E B2RXH2 3/20 0.47
MAPT P10636 3/20 0.47
LMNA P02545 3/20 0.47
POLB P06746 2/20 0.47
HSD17B10 Q99714 2/20 0.47
TP53 P04637 1/20 0.47
MEN1 O00255 1/20 0.44
GAA P10253 1/20 0.44
KMT2A Q03164 1/20 0.44
MAPK1 P28482 1/20 0.43
HTT P42858 1/20 0.43
GPR3 P46089 1/20 0.41
CDK5 Q00535 1/20 0.41
CDK5R1 Q15078 1/20 0.41
ALDH1A1 P00352 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9138426 0.79 HTR3E (0.52) HTR3EHTR3BHTR3AHTR3DHTR3C
SCHEMBL10099727 0.79 HTR3E (0.52) HTR3EHTR3BHTR3AHTR3DHTR3C
SCHEMBL9258182 0.75 HTR3E (0.49) HTR3EHTR3BHTR3AHTR3DHTR3C
SCHEMBL11326164 0.72 HTR3E (0.47) HTR3EHTR3BHTR3AHTR3DHTR3C
SCHEMBL363210 0.70 KDM4E (0.54) KDM4EMAPTLMNAPOLBHSD17B10
SCHEMBL3384231 0.70 HTR3E (0.42) HTR3EHTR3BHTR3AHTR3DHTR3C
SCHEMBL31461670 0.68 KDM4E (0.42) KDM4EMAPTLMNAPOLBHSD17B10
SCHEMBL31461727 0.68 TSHR (0.42) KDM4EMAPTLMNAPOLBHSD17B10
SCHEMBL11474094 0.68 ALOX15 (0.46) KDM4EMAPTLMNAPOLBHSD17B10
SCHEMBL11325773 0.68 MAPT (0.51) KDM4EMAPTLMNAPOLBHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012007006-A1 TRIAZOLO- AND PYRAZOLOQUINAZOLINE DERIVATIVES AS PDE10A ENZYME INHIBITOR H. LUNDBECK A/S (DK) 2012-01-19 WO disclosed