SCHEMBL363059

SCHEMBL363059

Cc1ccccc1[C@H](C/C(=N/O)c1c[nH]c(=O)c(C)c1)c1ccc(C#N)cc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GPBAR1 Q8TDU6 6/20 0.46
BRD4 O60885 1/20 0.37
CTSA P10619 4/20 0.35
MAPT P10636 2/20 0.35
L3MBTL1 Q9Y468 2/20 0.35
MEN1 O00255 1/20 0.35
ALDH1A1 P00352 1/20 0.35
KMT2A Q03164 1/20 0.35
MCL1 Q07820 1/20 0.35
PRSS1 P07477 1/20 0.34
CTSG P08311 1/20 0.34
CTRB1 P17538 1/20 0.34
CMA1 P23946 1/20 0.34
GAA P10253 2/20 0.33
KDM4E B2RXH2 1/20 0.33
TOP2A P11388 1/20 0.32
TOP2B Q02880 1/20 0.32
MGAM O43451 1/20 0.32
SI P14410 1/20 0.32
MGAM2 Q2M2H8 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL363163 1.00 GPBAR1 (0.46) GPBAR1BRD4CTSAMAPTL3MBTL1
SCHEMBL363678 0.87 GPBAR1 (0.61) GPBAR1BRD4CTSAL3MBTL1MEN1
SCHEMBL364664 0.87 GAA (0.42) GPBAR1BRD4CTSAMAPTL3MBTL1
SCHEMBL362796 0.85 GPBAR1 (0.39) GPBAR1BRD4CTSAMAPTL3MBTL1
SCHEMBL364092 0.84 GPBAR1 (0.48) GPBAR1BRD4CTSAGAAMGAM
SCHEMBL362545 0.84 GPBAR1 (0.66) GPBAR1BRD4CTSAGAAMGAM
SCHEMBL364601 0.84 GPBAR1 (0.66) GPBAR1BRD4CTSAGAAMGAM
SCHEMBL363349 0.84 GPBAR1 (0.66) GPBAR1BRD4CTSAGAAMGAM
SCHEMBL363650 0.82 GPBAR1 (0.58) GPBAR1BRD4CTSAGAAMGAM
SCHEMBL362350 0.81 GPBAR1 (0.48) GPBAR1BRD4CTSAMAPTKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2593426-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F.HOFFMANN-LA ROCHE AG (CH) 2013-05-22 EP claimed
WO-2012007365-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F. HOFFMANN-LA ROCHE AG (CH) 2012-01-19 WO claimed
EP-2593426-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F.HOFFMANN-LA ROCHE AG (CH) 2013-05-22 EP disclosed
WO-2012007365-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F. HOFFMANN-LA ROCHE AG (CH) 2012-01-19 WO disclosed