SCHEMBL364092

SCHEMBL364092

Cc1ccccc1[C@H](C/C(=N\O)c1c[nH]c(=O)c(C)c1)c1ccc(CC(=O)O)cc1

nearest known ligand 0.48

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
GPBAR1 Q8TDU6 6/20 0.48
BRD4 O60885 1/20 0.39
FFAR1 O14842 2/20 0.35
MGAM O43451 2/20 0.34
GAA P10253 2/20 0.34
SI P14410 2/20 0.34
MGAM2 Q2M2H8 2/20 0.34
CTSA P10619 4/20 0.33
NR3C2 P08235 1/20 0.32
LMNA P02545 1/20 0.32
TAAR1 Q96RJ0 1/20 0.32
SRD5A2 P31213 1/20 0.31
KEAP1 Q14145 1/20 0.31
NFE2L2 Q16236 1/20 0.31
MAPK1 P28482 1/20 0.31
NPSR1 Q6W5P4 1/20 0.31
CYP3A4 P08684 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL363678 0.89 GPBAR1 (0.61) GPBAR1BRD4MGAMGAASI
SCHEMBL361676 0.88 GPBAR1 (0.51) GPBAR1BRD4FFAR1CTSALMNA
SCHEMBL364841 0.88 GAA (0.43) GPBAR1BRD4FFAR1MGAMGAA
SCHEMBL363349 0.86 GPBAR1 (0.66) GPBAR1BRD4MGAMGAASI
SCHEMBL362545 0.86 GPBAR1 (0.66) GPBAR1BRD4MGAMGAASI
SCHEMBL364601 0.86 GPBAR1 (0.66) GPBAR1BRD4MGAMGAASI
Hydroxyamine SCHEMBL363012 0.86 GAA (0.41) GPBAR1BRD4FFAR1MGAMGAA
SCHEMBL362350 0.85 GPBAR1 (0.48) GPBAR1BRD4CTSACYP3A4
SCHEMBL363059 0.84 GPBAR1 (0.46) GPBAR1BRD4MGAMGAASI
SCHEMBL363163 0.84 GPBAR1 (0.46) GPBAR1BRD4MGAMGAASI

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2593426-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F.HOFFMANN-LA ROCHE AG (CH) 2013-05-22 EP claimed
WO-2012007365-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F. HOFFMANN-LA ROCHE AG (CH) 2012-01-19 WO claimed
EP-2593426-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F.HOFFMANN-LA ROCHE AG (CH) 2013-05-22 EP disclosed
WO-2012007365-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F. HOFFMANN-LA ROCHE AG (CH) 2012-01-19 WO disclosed